TY  - JOUR
AU  - Szatmári, István
AU  - Fülöp, Ferenc
TI  - Syntheses, transformations and applications of aminonaphthol derivatives prepared via modified Mannich reactions
JF  - TETRAHEDRON
J2  - TETRAHEDRON
VL  - 69
PY  - 2013
IS  - 4
SP  - 1255
EP  - 1278
PG  - 24
SN  - 0040-4020
DO  - 10.1016/j.tet.2012.11.055
UR  - https://m2.mtmt.hu/api/publication/2221504
ID  - 2221504
N1  - Cited By :61            
            Export Date: 15 October 2021            
            CODEN: TETRA            
            Correspondence Address: Fülöp, F.; Institute of Pharmaceutical Chemistry, Eötvös u. 6, H-6720 Szeged, Hungary; email: fulop@pharm.u-szeged.hu            
            Chemicals/CAS: imine, 13774-92-0
LA  - English
DB  - MTMT
ER  - 

TY  - JOUR
AU  - Szatmári, István
AU  - Fülöp, Ferenc
TI  - Simple access to pentacyclic oxazinoisoquinolines via an unexpected transformation of aminomethylnaphthols
JF  - TETRAHEDRON LETTERS
J2  - TETRAHEDRON LETT
VL  - 52
PY  - 2011
IS  - 34
SP  - 4440
EP  - 4442
PG  - 3
SN  - 0040-4039
DO  - 10.1016/j.tetlet.2011.06.074
UR  - https://m2.mtmt.hu/api/publication/1700166
ID  - 1700166
N1  - Cited By :22            
            Export Date: 15 October 2021            
            CODEN: TELEA            
            Correspondence Address: Fülöp, F.; Institute of Pharmaceutical Chemistry, Eötvös u. 6, H-6720 Szeged, Hungary; email: fulop@pharm.u-szeged.hu            
            Funding details: Hungarian Scientific Research Fund, K-75433, TÁMOP-4.2.1/B-09/1/KONV-2010-0005            
            Funding text 1: The authors thank the Hungarian Research Foundation (OTKA No. K-75433 ) and TÁMOP-4.2.1/B-09/1/KONV-2010-0005 for financial support. S.I. acknowledges the award of a Bolyai János Fellowship.
AB  - Unexpected reactions between 1-alpha-aminobenzyl-2-naphthol, 1-aminomethyl-2-naphthol, N-benzyl-1-alpha-aminobenzyl-2-naphthol and 6,7-dimethoxy-3,4-dihydroisoquinoline to furnish naphth[1,2-e][1,3]oxazino[2,3-a]isoquinolines are reported. The reaction conditions involved classical heating at 80 degrees C in MeCN for 22 h (57-62%), or the use of microwave conditions (100 degrees C), which allowed a reduction of the reaction time to 90 min and resulted in somewhat higher yields (73-82%). (C) 2011 Elsevier Ltd. All rights reserved.
LA  - English
DB  - MTMT
ER  - 

TY  - JOUR
AU  - Szatmári, István
AU  - Hetényi, Anasztázia
AU  - Lázár, László
AU  - Fülöp, Ferenc
TI  - Transformation reactions of the Betti base analog aminonaphthols
JF  - JOURNAL OF HETEROCYCLIC CHEMISTRY
J2  - J HETEROCYCLIC CHEM
VL  - 41
PY  - 2004
IS  - 3
SP  - 367
EP  - 373
PG  - 7
SN  - 0022-152X
DO  - 10.1002/jhet.5570410310
UR  - https://m2.mtmt.hu/api/publication/1013250
ID  - 1013250
AB  - By means of simple or domino ring-closure reactions of 1-(alpha-aminobenzyl)-2-naphthol (Betti base: 1), 1-aminomethyl-2-naplithol (2) and 2-(alpha-aminobenzyl)-1-naphthol (reverse Berri base: 3) with phosgene, ethyl benzimidate, 2-carboxybenzaldehyde, levulinic acid, salicylaldehyde/formalin or salicylaldehyde/acetaldehyde, naphth[1,2-e][1,3]oxazine and naphth[2,1-e][1,3]oxazine derivatives were prepared. All of the nitrogen-bridged polycyclic derivatives of 1 and 3 containing a number of centers of asymmetry were formed with nearly complete diastereoselectivity. Considerable differences were observed in the ring-closing abilities of the unsubstituted and phenyl-substituted aminonaphthols 1 and 2 and of the regioisomeric compounds 1 and 3.
LA  - English
DB  - MTMT
ER  -