TY - JOUR AU - Peřina, Miroslav AU - Kiss, Anita AU - Mernyák, Erzsébet AU - Mada, Lukáš AU - Schneider, Gyula AU - Jorda, Radek TI - Synthesis of hydrocortisone esters targeting androgen and glucocorticoid receptors in prostate cancer in vitro JF - JOURNAL OF STEROID BIOCHEMISTRY AND MOLECULAR BIOLOGY J2 - J STEROID BIOCHEM MOL BIOL VL - 229 PY - 2023 PG - 12 SN - 0960-0760 DO - 10.1016/j.jsbmb.2023.106269 UR - https://m2.mtmt.hu/api/publication/33663109 ID - 33663109 LA - English DB - MTMT ER - TY - JOUR AU - Kiss, Anita AU - Jójárt, Rebeka AU - Mernyák, Erzsébet AU - Bartha, Sándor AU - Minorics, Renáta AU - Zupkó, István AU - Schneider, Gyula TI - Novel preparation of substituted oxazolines condensed to d-ring of estrane skeleton and characterization of their antiproliferative properties JF - STEROIDS J2 - STEROIDS VL - 176 PY - 2021 PG - 6 SN - 0039-128X DO - 10.1016/j.steroids.2021.108911 UR - https://m2.mtmt.hu/api/publication/32241841 ID - 32241841 LA - English DB - MTMT ER - TY - JOUR AU - Nagymihaly, Zoltan AU - Wölfling, János AU - Schneider, Gyula AU - Kollár, László TI - Synthesis of 2‐Methylresorcinol‐Based Deepened Cavitands with Chiral Inlet Bearing Steroidal Moieties on the Upper Rim JF - CHEMISTRYSELECT J2 - CHEMISTRYSELECT VL - 5 PY - 2020 IS - 23 SP - 6933 EP - 6938 PG - 6 SN - 2365-6549 DO - 10.1002/slct.202001728 UR - https://m2.mtmt.hu/api/publication/31355906 ID - 31355906 N1 - Funding Agency and Grant Number: Hungarian Scientific Research Fund [OTKA K113177]; Ultrafast physical processes in atom, molecules, nanostructures and biological systems [EFOP-3.6.2-16-2017-00005]; [GINOP-2.3.2-15-2016-00049] Funding text: The authors thank the Hungarian Scientific Research Fund (OTKA K113177) for the financial support and Johnson Matthey for the generous gift of palladium(II) acetate. This work was supported by the GINOP-2.3.2-15-2016-00049 grant. Financial support from the Ultrafast physical processes in atom, molecules, nanostructures and biological systems (EFOP-3.6.2-16-2017-00005) is gratefully acknowledged. LA - English DB - MTMT ER - TY - JOUR AU - Kiss, Anita AU - Wölfling, János AU - Mernyák, Erzsébet AU - Nagyné Frank, Éva AU - Benke, Zsanett Amália AU - Senobar Tahaei, Seyyed Ashkan AU - Zupkó, István AU - Mahó, Sándor AU - Schneider, Gyula TI - Stereocontrolled synthesis of the four possible 3-methoxy and 3-benzyloxy-16-triazolyl-methyl-estra-17-ol hybrids and their antiproliferative activities JF - STEROIDS J2 - STEROIDS VL - 152 PY - 2019 PG - 14 SN - 0039-128X DO - 10.1016/j.steroids.2019.108500 UR - https://m2.mtmt.hu/api/publication/30838971 ID - 30838971 N1 - Department of Organic Chemistry, University of Szeged, Dóm tér 8, H-6720 Szeged, Hungary Institute of Pharmaceutical Chemistry, University of Szeged, H-6720, Eötvös u. 6, H-6720 Szeged, Hungary Department of Pharmacodynamics and Biopharmacy, University of Szeged, Eötvös u. 6, H-6720 Szeged, Hungary Interdisciplinary Centre for Natural Products, University of Szeged, Eötvös u. 6, H-6720 Szeged, Hungary Chemical Works of Gedeon Richter Plc., Gyömrői út 19-21, H-1103 Budapest, Hungary Export Date: 11 February 2020 CODEN: STEDA Correspondence Address: Schneider, G.; Department of Organic Chemistry, University of Szeged, Dóm tér 8, Hungary; email: schneider@chem.u-szeged.hu Chemicals/CAS: cisplatin, 15663-27-1, 26035-31-4, 96081-74-2 Funding details: Emberi Eroforrások Minisztériuma, 20391-3/2018/FEKUSTRAT Funding details: Hungarian Scientific Research Fund, OTKA Funding details: GINOP-2.3.2-15-2016-00038, EFOP-3.6.2 Funding details: Richter Gedeon Talentum Alapítvány Funding details: K113150 Funding text 1: The work of Anita Kiss was supported by a PhD Fellowship of the Talentum Fund of Richter Gedeon Plc. (Budapest). Financial support from the Economic Development and Innovation Operative Programme of Hungary (GINOP-2.3.2-15-2016-00038) and Ultrafast physical processes in atoms, molecules, nanostructures and biological systems (No: EFOP-3.6.2.-2017-00005) is gratefully acknowledged. This research was supported by the Hungarian Scientific Research Fund (OTKA K113150 ). Ministry of Human Capacities , Hungary grant 20391-3/2018/FEKUSTRAT is acknowledged. Appendix A Funding Agency and Grant Number: Talentum Fund of Richter Gedeon Plc. (Budapest); Economic Development and Innovation Operative Programme of Hungary [GINOP-2.3.2-15-2016-00038]; Ultrafast physical processes in atoms, molecules, nanostructures and biological systems [EFOP-3.6.2.-2017-00005]; Hungarian Scientific Research Fund, Ministry of Human Capacities, Hungary [OTKA K113150, 20391-3/2018/FEKUSTRAT] Funding text: The work of Anita Kiss was supported by a PhD Fellowship of the Talentum Fund of Richter Gedeon Plc. (Budapest). Financial support from the Economic Development and Innovation Operative Programme of Hungary (GINOP-2.3.2-15-2016-00038) and Ultrafast physical processes in atoms, molecules, nanostructures and biological systems (No: EFOP-3.6.2.-2017-00005) is gratefully acknowledged. This research was supported by the Hungarian Scientific Research Fund (OTKA K113150). Ministry of Human Capacities, Hungary grant 20391-3/2018/FEKUSTRAT is acknowledged. Department of Organic Chemistry, University of Szeged, Dóm tér 8, H-6720 Szeged, Hungary Institute of Pharmaceutical Chemistry, University of Szeged, H-6720, Eötvös u. 6, H-6720 Szeged, Hungary Department of Pharmacodynamics and Biopharmacy, University of Szeged, Eötvös u. 6, H-6720 Szeged, Hungary Interdisciplinary Centre for Natural Products, University of Szeged, Eötvös u. 6, H-6720 Szeged, Hungary Chemical Works of Gedeon Richter Plc., Gyömrői út 19-21, H-1103 Budapest, Hungary Cited By :1 Export Date: 29 August 2020 CODEN: STEDA Correspondence Address: Schneider, G.; Department of Organic Chemistry, University of Szeged, Dóm tér 8, Hungary; email: schneider@chem.u-szeged.hu Chemicals/CAS: cisplatin, 15663-27-1, 26035-31-4, 96081-74-2; Antineoplastic Agents; Triazoles Funding details: Emberi Eroforrások Minisztériuma, 20391-3/2018/FEKUSTRAT Funding details: Hungarian Scientific Research Fund, OTKA Funding details: GINOP-2.3.2-15-2016-00038, EFOP-3.6.2 Funding details: Richter Gedeon Talentum Alapítvány Funding details: K113150 Funding text 1: The work of Anita Kiss was supported by a PhD Fellowship of the Talentum Fund of Richter Gedeon Plc. (Budapest). Financial support from the Economic Development and Innovation Operative Programme of Hungary (GINOP-2.3.2-15-2016-00038) and Ultrafast physical processes in atoms, molecules, nanostructures and biological systems (No: EFOP-3.6.2.-2017-00005) is gratefully acknowledged. This research was supported by the Hungarian Scientific Research Fund (OTKA K113150 ). Ministry of Human Capacities , Hungary grant 20391-3/2018/FEKUSTRAT is acknowledged. Appendix A Department of Organic Chemistry, University of Szeged, Dóm tér 8, H-6720 Szeged, Hungary Institute of Pharmaceutical Chemistry, University of Szeged, H-6720, Eötvös u. 6, H-6720 Szeged, Hungary Department of Pharmacodynamics and Biopharmacy, University of Szeged, Eötvös u. 6, H-6720 Szeged, Hungary Interdisciplinary Centre for Natural Products, University of Szeged, Eötvös u. 6, H-6720 Szeged, Hungary Chemical Works of Gedeon Richter Plc., Gyömrői út 19-21, H-1103 Budapest, Hungary Cited By :1 Export Date: 10 January 2021 CODEN: STEDA Correspondence Address: Schneider, G.; Department of Organic Chemistry, University of Szeged, Dóm tér 8, Hungary; email: schneider@chem.u-szeged.hu Chemicals/CAS: cisplatin, 15663-27-1, 26035-31-4, 96081-74-2; Antineoplastic Agents; Triazoles Funding details: Emberi Eroforrások Minisztériuma, EMMI, 20391-3/2018/FEKUSTRAT Funding details: Hungarian Scientific Research Fund, OTKA, OTKA K113150 Funding details: Richter Gedeon Talentum Alapítvány Funding details: -2017-00005, GINOP-2.3.2-15-2016-00038, EFOP-3.6.2 Funding text 1: The work of Anita Kiss was supported by a PhD Fellowship of the Talentum Fund of Richter Gedeon Plc. (Budapest). Financial support from the Economic Development and Innovation Operative Programme of Hungary (GINOP-2.3.2-15-2016-00038) and Ultrafast physical processes in atoms, molecules, nanostructures and biological systems (No: EFOP-3.6.2.-2017-00005) is gratefully acknowledged. This research was supported by the Hungarian Scientific Research Fund (OTKA K113150 ). Ministry of Human Capacities , Hungary grant 20391-3/2018/FEKUSTRAT is acknowledged. LA - English DB - MTMT ER - TY - JOUR AU - Herman, Bianka Edina AU - Kiss, Anita AU - Wölfling, János AU - Mernyák, Erzsébet AU - Szécsi, Mihály AU - Schneider, Gyula TI - Synthesis of substituted 15β-alkoxy estrone derivatives and their cofactor-dependent inhibitory effect on 17β-HSD1 JF - JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY J2 - J ENZYM INHIB MED CH VL - 34 PY - 2019 IS - 1 SP - 1271 EP - 1286 PG - 16 SN - 1475-6366 DO - 10.1080/14756366.2019.1634064 UR - https://m2.mtmt.hu/api/publication/30747981 ID - 30747981 N1 - Export Date: 6 August 2019 LA - English DB - MTMT ER - TY - JOUR AU - Kiss, Anita AU - Wölfling, János AU - Mernyák, Erzsébet AU - Nagyné Frank, Éva AU - Gyovai, András AU - Kulmány, Ágnes Erika AU - Zupkó, István AU - Schneider, Gyula TI - Stereoselective Synthesis of New Type of Estradiol Hybrid Molecules and their Antiproliferative Activities JF - STEROIDS J2 - STEROIDS VL - 148 PY - 2019 SP - 63 EP - 72 PG - 10 SN - 0039-128X DO - 10.1016/j.steroids.2019.02.016 UR - https://m2.mtmt.hu/api/publication/30672538 ID - 30672538 LA - English DB - MTMT ER - TY - JOUR AU - Jójárt, Rebeka AU - Traj, Péter AU - Kovács, Édua AU - Horváth, Ágnes AU - Schneider, Gyula AU - Szécsi, Mihály AU - Pál, Attila AU - Paragi, Gábor AU - Mernyák, Erzsébet TI - Synthesis, Biological Evaluation and Docking Studies of 13-Epimeric 10-fluoro- and 10-Chloroestra-1,4-dien-3-ones as Potential Aromatase Inhibitors JF - MOLECULES J2 - MOLECULES VL - 24 PY - 2019 IS - 9 PG - 18 SN - 1420-3049 DO - 10.3390/molecules24091783 UR - https://m2.mtmt.hu/api/publication/30672179 ID - 30672179 N1 - WoS:hiba:000469518100142 2020-01-10 07:35 cikkazonosító nem egyezik LA - English DB - MTMT ER - TY - JOUR AU - Jopp, Stefan AU - Ehlers, Peter AU - Nagyné Frank, Éva AU - Mernyák, Erzsébet AU - Schneider, Gyula AU - Wölfling, János AU - Villinger, Alexander AU - Langer, Peter TI - Site-Selective Synthesis of 3,17-Diaryl-1,3,5,16-estratetraenes JF - SYNLETT J2 - SYNLETT VL - 30 ET - 0 PY - 2019 IS - 5 SP - 600 EP - 604 PG - 5 SN - 0936-5214 DO - 10.1055/s-0037-1611720 UR - https://m2.mtmt.hu/api/publication/30429176 ID - 30429176 LA - English DB - MTMT ER - TY - JOUR AU - Froehlich, Tony AU - Kiss, Anita AU - Wölfling, János AU - Mernyák, Erzsébet AU - Kulmány, Ágnes Erika AU - Minorics, Renáta AU - Zupkó, István AU - Leidenberger, Maria AU - Friedrich, Oliver AU - Kappes, Barbara AU - Hahn, Friedrich AU - Marschall, Manfred AU - Schneider, Gyula AU - Tsogoeva, Svetlana B. TI - Synthesis of Artemisinin-Estrogen Hybrids Highly Active against HCMV, P. falciparum, and Cervical and Breast Cancer JF - ACS MEDICINAL CHEMISTRY LETTERS J2 - ACS MED CHEM LETT VL - 9 PY - 2018 IS - 11 SP - 1128 EP - 1133 PG - 6 SN - 1948-5875 DO - 10.1021/acsmedchemlett.8b00381 UR - https://m2.mtmt.hu/api/publication/30387211 ID - 30387211 LA - English DB - MTMT ER - TY - JOUR AU - Bacsa, Ildikó AU - Herman, Bianka Edina AU - Jójárt, Rebeka AU - Herman, Kevin Stefan AU - Wölfling, János AU - Schneider, Gyula AU - Varga, Mónika AU - Tömböly, Csaba AU - Rizner, Tea Lanisnik AU - Szécsi, Mihály AU - Mernyák, Erzsébet TI - Synthesis and structure–activity relationships of 2- and/or 4-halogenated 13β- and 13α-estrone derivatives as enzyme inhibitors of estrogen biosynthesis JF - JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY J2 - J ENZYM INHIB MED CH VL - 33 PY - 2018 IS - 1 SP - 1271 EP - 1282 PG - 12 SN - 1475-6366 DO - 10.1080/14756366.2018.1490731 UR - https://m2.mtmt.hu/api/publication/27701563 ID - 27701563 N1 - Department of Organic Chemistry, University of Szeged, Szeged, Hungary 1st Department of Medicine, University of Szeged, Szeged, Hungary Department of Microbiology, University of Szeged, University of Szeged, Szeged, Hungary Laboratory of Chemical Biology, Institute of Biochemistry, Biological Research Centre of the Hungarian Academy of Sciences, Szeged, Hungary Institute of Biochemistry, Faculty of Medicine, University of Ljubljana, Ljubljana, Slovenia Cited By :19 Export Date: 3 May 2022 CODEN: JEIMA Correspondence Address: Mernyák, E.; Department of Organic Chemistry, Dóm tér 8, Hungary; email: bobe@chem.u-szeged.hu Chemicals/CAS: aromatase, 9039-48-9; hydroxysteroid dehydrogenase, 9001-56-3; steryl sulfatase, 9025-62-1; estradiol 17beta dehydrogenase, 9028-61-9; estrone, 53-16-7; Aromatase; Enzyme Inhibitors; Estradiol Dehydrogenases; Estrogens; Estrone; HSD17B1 protein, human; Steryl-Sulfatase LA - English DB - MTMT ER -