@article{MTMT:30747981,
	author = {Herman, Bianka Edina and Kiss, Anita and Wölfling, János and Mernyák, Erzsébet and Szécsi, Mihály and Schneider, Gyula},
	doi = {10.1080/14756366.2019.1634064},
	title = {Synthesis of substituted 15β-alkoxy estrone derivatives and their cofactor-dependent inhibitory effect on 17β-HSD1},
	journal-iso = {J ENZYM INHIB MED CH},
	journal = {JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY},
	volume = {34},
	unique-id = {30747981},
	issn = {1475-6366},
	year = {2019},
	pages = {1271-1286},
	orcid-numbers = {Wölfling, János/0000-0002-3037-309X; Mernyák, Erzsébet/0000-0003-4494-1817}
}

@article{MTMT:30672179,
	author = {Jójárt, Rebeka and Traj, Péter and Kovács, Édua and Horváth, Ágnes and Schneider, Gyula and Szécsi, Mihály and Pál, Attila and Paragi, Gábor and Mernyák, Erzsébet},
	doi = {10.3390/molecules24091783},
	title = {Synthesis, Biological Evaluation and Docking Studies of 13-Epimeric 10-fluoro- and 10-Chloroestra-1,4-dien-3-ones as Potential Aromatase Inhibitors},
	journal-iso = {MOLECULES},
	journal = {MOLECULES},
	volume = {24},
	unique-id = {30672179},
	issn = {1420-3049},
	year = {2019},
	orcid-numbers = {Paragi, Gábor/0000-0001-5408-1748; Mernyák, Erzsébet/0000-0003-4494-1817}
}

@CONFERENCE{MTMT:30462098,
	author = {Jójárt, R and Pécsy, Sz and Szlávik, M and Szabó, V and Traj, P and Szécsi, Mihály and Rigó, R and Özvegy-Laczka, Cs and Mernyák, E},
	booktitle = {Serbian Biochemical Society - Eighth Conference},
	title = {Synthesis and biochemical evaluation of novel 13?-estrone derivatives for targeted intracrine modulation of estrogen biosynthesis and transport},
	unique-id = {30462098},
	year = {2018},
	pages = {137-138}
}

@{MTMT:30462091,
	author = {Jovanović-Šanta, SS and Herman, Bianka Edina and Zupkó, István and Kulmány, Ágnes Erika and Zupkó, István and Nikolić, AR and Savić, M and Oklješa, A and Szécsi, Mihály},
	booktitle = {FEBS3+ Conference; From molecules to living systems},
	title = {Screening of Antihormonal and Anticancer Potential of Heterocyclic Estrane Steroids},
	unique-id = {30462091},
	year = {2018},
	pages = {247},
	orcid-numbers = {Zupkó, István/0000-0003-3243-5300; Zupkó, István/0000-0003-3243-5300}
}

@article{MTMT:30331520,
	author = {Jójárt, Rebeka and Pécsy, S. and Keglevich, György and Szécsi, Mihály and Rigó, R. and Laczka, Csilla and Kecskeméti, Gábor and Mernyák, Erzsébet},
	doi = {10.3762/bjoc.14.262},
	title = {Pd-Catalyzed microwave-assisted synthesis of phosphonated 13α-estrones as potential OATP2B1, 17β-HSD1 and/or STS inhibitors},
	journal-iso = {BEILSTEIN J ORG CHEM},
	journal = {BEILSTEIN JOURNAL OF ORGANIC CHEMISTRY},
	volume = {14},
	unique-id = {30331520},
	issn = {1860-5397},
	abstract = {Novel 2- or 4-phosphonated 13 alpha-estrone derivatives were synthesized via the Hirao reaction. Bromo regioisomers (2- or 4-) of 13 alpha-estrone and its 3-benzyl or 3-methyl ether were reacted with diethyl phosphite or diphenylphosphine oxide using Pd(PPh3)(4) as catalyst under microwave irradiation. The influence of the new compounds on the transport function of the organic anion transporting polypeptide OATP2B1 was investigated by measuring Cascade Blue uptake. Derivatives bearing a 3-benzyl ether function displayed substantial submicromolar OATP2B1 inhibitory activity. The inhibitory effects of the compounds on human placental steroid sulfatase (STS) and 17 beta-hydroxysteroid dehydrogenase type 1 isozyme (17 beta-HSD1) were investigated by in vitro radiosub-strate incubation methods. None of the test compounds inhibited the STS markedly. The structure-activity relationship evaluation revealed that 2-substituted 3-hydroxy derivatives are able to inhibit the 17 beta-HSD1 enzyme with submicromolar IC50 values. Dual OATP2B1 and 17 beta-HSD1 inhibitors have been identified.},
	keywords = {ENZYME; CATALYSIS; STS; Hirao reaction; OATP2B1; 13 alpha-estrone; 17 beta-HSD1 inhibition},
	year = {2018},
	pages = {2838-2845},
	orcid-numbers = {Mernyák, Erzsébet/0000-0003-4494-1817}
}

@article{MTMT:27701563,
	author = {Bacsa, Ildikó and Herman, Bianka Edina and Jójárt, Rebeka and Herman, Kevin Stefan and Wölfling, János and Schneider, Gyula and Varga, Mónika and Tömböly, Csaba and Rizner, Tea Lanisnik and Szécsi, Mihály and Mernyák, Erzsébet},
	doi = {10.1080/14756366.2018.1490731},
	title = {Synthesis and structure–activity relationships of 2- and/or 4-halogenated 13β- and 13α-estrone derivatives as enzyme inhibitors of estrogen biosynthesis},
	journal-iso = {J ENZYM INHIB MED CH},
	journal = {JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY},
	volume = {33},
	unique-id = {27701563},
	issn = {1475-6366},
	year = {2018},
	pages = {1271-1282},
	orcid-numbers = {Bacsa, Ildikó/0000-0001-8277-631X; Wölfling, János/0000-0002-3037-309X; Mernyák, Erzsébet/0000-0003-4494-1817}
}

@article{MTMT:3372993,
	author = {Kiss, Anita and Herman, Bianka Edina and Görbe, Tamás and Mernyák, Erzsébet and Molnár, Barnabás and Wölfling, János and Szécsi, Mihály and Schneider, Gyula},
	doi = {10.1016/j.steroids.2018.03.006},
	title = {Synthesis of novel 17-triazolyl-androst-5-en-3-ol epimers via Cu(I)-catalyzed azide-alkyne cycloaddition and their inhibitory effect on 17α-hydroxylase/C17,20-lyase},
	journal-iso = {STEROIDS},
	journal = {STEROIDS},
	volume = {135},
	unique-id = {3372993},
	issn = {0039-128X},
	year = {2018},
	eissn = {1878-5867},
	pages = {79-91},
	orcid-numbers = {Mernyák, Erzsébet/0000-0003-4494-1817; Wölfling, János/0000-0002-3037-309X}
}

@article{MTMT:3251236,
	author = {Bacsa, Ildikó and Jójárt, Rebeka and Wölfling, János and Schneider, Gyula and Herman, Bianka Edina and Szécsi, Mihály and Mernyák, Erzsébet},
	doi = {10.3762/bjoc.13.126},
	title = {Synthesis of novel 13 alpha-estrone derivatives by Sonogashira coupling as potential 17 beta-HSD1 inhibitors},
	journal-iso = {BEILSTEIN J ORG CHEM},
	journal = {BEILSTEIN JOURNAL OF ORGANIC CHEMISTRY},
	volume = {13},
	unique-id = {3251236},
	issn = {1860-5397},
	year = {2017},
	pages = {1303-1309},
	orcid-numbers = {Bacsa, Ildikó/0000-0001-8277-631X; Wölfling, János/0000-0002-3037-309X; Mernyák, Erzsébet/0000-0003-4494-1817}
}

@article{MTMT:3227244,
	author = {Szánti-Pintér, Eszter and L, Maksó and Gömöry, Ágnes and J, Wouters and Herman, Bianka Edina and Szécsi, Mihály and Mikle, Gábor and Kollár, László and Skodáné Földes, Rita},
	doi = {10.1016/j.steroids.2017.05.006},
	title = {Synthesis of 16α-amino-pregnenolone derivatives via ionic liquid-catalyzed aza-Michael addition and their evaluation as C17,20-lyase inhibitors},
	journal-iso = {STEROIDS},
	journal = {STEROIDS},
	volume = {123},
	unique-id = {3227244},
	issn = {0039-128X},
	year = {2017},
	eissn = {1878-5867},
	pages = {61-66}
}

@article{MTMT:2939481,
	author = {Szabó, Johanna and Bacsa, Ildikó and Wölfling, János and Schneider, Gyula and Zupkó, István and Varga, Mónika and Herman, Bianka Edina and Kalmár, László and Szécsi, Mihály and Mernyák, Erzsébet},
	doi = {10.3109/14756366.2015.1050008},
	title = {Synthesis and in vitro pharmacological evaluation of N-[(1-benzyl-1,2,3-triazol-4-yl)methyl]-carboxamides on d-secoestrone scaffolds},
	journal-iso = {J ENZYM INHIB MED CH},
	journal = {JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY},
	volume = {31},
	unique-id = {2939481},
	issn = {1475-6366},
	year = {2016},
	pages = {574-579},
	orcid-numbers = {Bacsa, Ildikó/0000-0001-8277-631X; Wölfling, János/0000-0002-3037-309X; Zupkó, István/0000-0003-3243-5300; Mernyák, Erzsébet/0000-0003-4494-1817}
}