TY - JOUR AU - Wölfling, János TI - Schneider Gyula (1931–2021) JF - MAGYAR KÉMIKUSOK LAPJA J2 - MAGY KEM LAP VL - 77 PY - 2022 IS - 2 SP - 59 EP - 60 PG - 2 SN - 0025-0163 UR - https://m2.mtmt.hu/api/publication/33098465 ID - 33098465 LA - Hungarian DB - MTMT ER - TY - JOUR AU - Kovács, Attila AU - Csutorás, Csaba AU - Rajkó, Róbert AU - Sziva, Miklós AU - Wölfling, János TI - Közhasznúsági jelentés. a Magyar Kémikusok Egyesülete (MKE) 2019. évi közhasznú tevékenységéről és előterjesztés a 2020. évi terv főbb mutatóiról TS - a Magyar Kémikusok Egyesülete (MKE) 2019. évi közhasznú tevékenységéről és előterjesztés a 2020. évi terv főbb mutatóiról JF - MAGYAR KÉMIKUSOK LAPJA J2 - MAGY KEM LAP VL - 75 PY - 2020 IS - 11 SP - 323 EP - 330 PG - 8 SN - 0025-0163 UR - https://m2.mtmt.hu/api/publication/31810109 ID - 31810109 LA - Hungarian DB - MTMT ER - TY - JOUR AU - Angyal, Anikó AU - Demjen, Andras AU - Wölfling, János AU - Puskas, Laszlo G. AU - Kanizsai, Iván TI - Acid-Catalyzed 1,3-Dipolar Cycloaddition of 2H-Azirines with Nitrones: An Unexpected Access to 1,2,4,5-Tetrasubstituted Imidazoles JF - JOURNAL OF ORGANIC CHEMISTRY J2 - J ORG CHEM VL - 85 PY - 2020 IS - 5 SP - 3587 EP - 3595 PG - 9 SN - 0022-3263 DO - 10.1021/acs.joc.9b03288 UR - https://m2.mtmt.hu/api/publication/31499509 ID - 31499509 AB - The first 1,3-dipolar cycloaddition of 2H-azirines with nitrones, a straightforward approach toward the regioselective synthesis of 1,2,4,5-tetrasubstituted imidazoles, is reported. This trifluoroacetic acid-catalyzed protocol tolerates a broad range of aliphatic and aromatic substrates, offering an efficient access to highly diverse, multisubstituted imidazoles in isolated yields up to 83% under mild conditions. LA - English DB - MTMT ER - TY - JOUR AU - Nagymihaly, Zoltan AU - Wölfling, János AU - Schneider, Gyula AU - Kollár, László TI - Synthesis of 2‐Methylresorcinol‐Based Deepened Cavitands with Chiral Inlet Bearing Steroidal Moieties on the Upper Rim JF - CHEMISTRYSELECT J2 - CHEMISTRYSELECT VL - 5 PY - 2020 IS - 23 SP - 6933 EP - 6938 PG - 6 SN - 2365-6549 DO - 10.1002/slct.202001728 UR - https://m2.mtmt.hu/api/publication/31355906 ID - 31355906 N1 - Funding Agency and Grant Number: Hungarian Scientific Research Fund [OTKA K113177]; Ultrafast physical processes in atom, molecules, nanostructures and biological systems [EFOP-3.6.2-16-2017-00005]; [GINOP-2.3.2-15-2016-00049] Funding text: The authors thank the Hungarian Scientific Research Fund (OTKA K113177) for the financial support and Johnson Matthey for the generous gift of palladium(II) acetate. This work was supported by the GINOP-2.3.2-15-2016-00049 grant. Financial support from the Ultrafast physical processes in atom, molecules, nanostructures and biological systems (EFOP-3.6.2-16-2017-00005) is gratefully acknowledged. LA - English DB - MTMT ER - TY - JOUR AU - Kiss, Anita AU - Wölfling, János AU - Mernyák, Erzsébet AU - Nagyné Frank, Éva AU - Benke, Zsanett Amália AU - Senobar Tahaei, Seyyed Ashkan AU - Zupkó, István AU - Mahó, Sándor AU - Schneider, Gyula TI - Stereocontrolled synthesis of the four possible 3-methoxy and 3-benzyloxy-16-triazolyl-methyl-estra-17-ol hybrids and their antiproliferative activities JF - STEROIDS J2 - STEROIDS VL - 152 PY - 2019 PG - 14 SN - 0039-128X DO - 10.1016/j.steroids.2019.108500 UR - https://m2.mtmt.hu/api/publication/30838971 ID - 30838971 N1 - Department of Organic Chemistry, University of Szeged, Dóm tér 8, H-6720 Szeged, Hungary Institute of Pharmaceutical Chemistry, University of Szeged, H-6720, Eötvös u. 6, H-6720 Szeged, Hungary Department of Pharmacodynamics and Biopharmacy, University of Szeged, Eötvös u. 6, H-6720 Szeged, Hungary Interdisciplinary Centre for Natural Products, University of Szeged, Eötvös u. 6, H-6720 Szeged, Hungary Chemical Works of Gedeon Richter Plc., Gyömrői út 19-21, H-1103 Budapest, Hungary Export Date: 11 February 2020 CODEN: STEDA Correspondence Address: Schneider, G.; Department of Organic Chemistry, University of Szeged, Dóm tér 8, Hungary; email: schneider@chem.u-szeged.hu Chemicals/CAS: cisplatin, 15663-27-1, 26035-31-4, 96081-74-2 Funding details: Emberi Eroforrások Minisztériuma, 20391-3/2018/FEKUSTRAT Funding details: Hungarian Scientific Research Fund, OTKA Funding details: GINOP-2.3.2-15-2016-00038, EFOP-3.6.2 Funding details: Richter Gedeon Talentum Alapítvány Funding details: K113150 Funding text 1: The work of Anita Kiss was supported by a PhD Fellowship of the Talentum Fund of Richter Gedeon Plc. (Budapest). Financial support from the Economic Development and Innovation Operative Programme of Hungary (GINOP-2.3.2-15-2016-00038) and Ultrafast physical processes in atoms, molecules, nanostructures and biological systems (No: EFOP-3.6.2.-2017-00005) is gratefully acknowledged. This research was supported by the Hungarian Scientific Research Fund (OTKA K113150 ). Ministry of Human Capacities , Hungary grant 20391-3/2018/FEKUSTRAT is acknowledged. Appendix A Funding Agency and Grant Number: Talentum Fund of Richter Gedeon Plc. (Budapest); Economic Development and Innovation Operative Programme of Hungary [GINOP-2.3.2-15-2016-00038]; Ultrafast physical processes in atoms, molecules, nanostructures and biological systems [EFOP-3.6.2.-2017-00005]; Hungarian Scientific Research Fund, Ministry of Human Capacities, Hungary [OTKA K113150, 20391-3/2018/FEKUSTRAT] Funding text: The work of Anita Kiss was supported by a PhD Fellowship of the Talentum Fund of Richter Gedeon Plc. (Budapest). Financial support from the Economic Development and Innovation Operative Programme of Hungary (GINOP-2.3.2-15-2016-00038) and Ultrafast physical processes in atoms, molecules, nanostructures and biological systems (No: EFOP-3.6.2.-2017-00005) is gratefully acknowledged. This research was supported by the Hungarian Scientific Research Fund (OTKA K113150). Ministry of Human Capacities, Hungary grant 20391-3/2018/FEKUSTRAT is acknowledged. Department of Organic Chemistry, University of Szeged, Dóm tér 8, H-6720 Szeged, Hungary Institute of Pharmaceutical Chemistry, University of Szeged, H-6720, Eötvös u. 6, H-6720 Szeged, Hungary Department of Pharmacodynamics and Biopharmacy, University of Szeged, Eötvös u. 6, H-6720 Szeged, Hungary Interdisciplinary Centre for Natural Products, University of Szeged, Eötvös u. 6, H-6720 Szeged, Hungary Chemical Works of Gedeon Richter Plc., Gyömrői út 19-21, H-1103 Budapest, Hungary Cited By :1 Export Date: 29 August 2020 CODEN: STEDA Correspondence Address: Schneider, G.; Department of Organic Chemistry, University of Szeged, Dóm tér 8, Hungary; email: schneider@chem.u-szeged.hu Chemicals/CAS: cisplatin, 15663-27-1, 26035-31-4, 96081-74-2; Antineoplastic Agents; Triazoles Funding details: Emberi Eroforrások Minisztériuma, 20391-3/2018/FEKUSTRAT Funding details: Hungarian Scientific Research Fund, OTKA Funding details: GINOP-2.3.2-15-2016-00038, EFOP-3.6.2 Funding details: Richter Gedeon Talentum Alapítvány Funding details: K113150 Funding text 1: The work of Anita Kiss was supported by a PhD Fellowship of the Talentum Fund of Richter Gedeon Plc. (Budapest). Financial support from the Economic Development and Innovation Operative Programme of Hungary (GINOP-2.3.2-15-2016-00038) and Ultrafast physical processes in atoms, molecules, nanostructures and biological systems (No: EFOP-3.6.2.-2017-00005) is gratefully acknowledged. This research was supported by the Hungarian Scientific Research Fund (OTKA K113150 ). Ministry of Human Capacities , Hungary grant 20391-3/2018/FEKUSTRAT is acknowledged. Appendix A Department of Organic Chemistry, University of Szeged, Dóm tér 8, H-6720 Szeged, Hungary Institute of Pharmaceutical Chemistry, University of Szeged, H-6720, Eötvös u. 6, H-6720 Szeged, Hungary Department of Pharmacodynamics and Biopharmacy, University of Szeged, Eötvös u. 6, H-6720 Szeged, Hungary Interdisciplinary Centre for Natural Products, University of Szeged, Eötvös u. 6, H-6720 Szeged, Hungary Chemical Works of Gedeon Richter Plc., Gyömrői út 19-21, H-1103 Budapest, Hungary Cited By :1 Export Date: 10 January 2021 CODEN: STEDA Correspondence Address: Schneider, G.; Department of Organic Chemistry, University of Szeged, Dóm tér 8, Hungary; email: schneider@chem.u-szeged.hu Chemicals/CAS: cisplatin, 15663-27-1, 26035-31-4, 96081-74-2; Antineoplastic Agents; Triazoles Funding details: Emberi Eroforrások Minisztériuma, EMMI, 20391-3/2018/FEKUSTRAT Funding details: Hungarian Scientific Research Fund, OTKA, OTKA K113150 Funding details: Richter Gedeon Talentum Alapítvány Funding details: -2017-00005, GINOP-2.3.2-15-2016-00038, EFOP-3.6.2 Funding text 1: The work of Anita Kiss was supported by a PhD Fellowship of the Talentum Fund of Richter Gedeon Plc. (Budapest). Financial support from the Economic Development and Innovation Operative Programme of Hungary (GINOP-2.3.2-15-2016-00038) and Ultrafast physical processes in atoms, molecules, nanostructures and biological systems (No: EFOP-3.6.2.-2017-00005) is gratefully acknowledged. This research was supported by the Hungarian Scientific Research Fund (OTKA K113150 ). Ministry of Human Capacities , Hungary grant 20391-3/2018/FEKUSTRAT is acknowledged. LA - English DB - MTMT ER - TY - JOUR AU - Keglevich, András Imre AU - Zsiros, V. AU - Keglevich, Péter AU - Szigetvári, Á. AU - Dékány, M. AU - Szántay, Csaba (Ifj.) AU - Mernyák, Erzsébet AU - Wölfling, János AU - Hazai, László TI - Synthesis and in vitro antitumor effect of new vindoline-steroid hybrids JF - CURRENT ORGANIC CHEMISTRY J2 - CURR ORG CHEM VL - 23 PY - 2019 IS - 8 SP - 959 EP - 967 PG - 9 SN - 1385-2728 DO - 10.2174/1385272823666190614113218 UR - https://m2.mtmt.hu/api/publication/30792667 ID - 30792667 N1 - Export Date: 8 September 2019 Funding Agency and Grant Number: Hungarian Scientific Research Fund [OTKA K113150] Funding text: This project was supported by the Hungarian Scientific Research Fund (OTKA K113150). Department of Organic Chemistry and Technology, Budapest University of Technology and Economics, Gellért tér 4, Budapest, H-1111, Hungary Quality Process Development Department, Egis Pharmaceuticals Plc, Keresztúri út 30-38, Budapest, H-1106, Hungary Spectroscopic Research Department, Gedeon Richter Plc, 10, P. O. Box 27, Budapest, H-1475, Hungary Department of Organic Chemistry, University of Szeged, Dóm tér 8, Szeged, H-6720, Hungary Cited By :1 Export Date: 16 May 2021 CODEN: CORCF Correspondence Address: Keglevich, P.; Department of Organic Chemistry and Technology, Gellért tér 4, Hungary; email: pkeglevich@mail.bme.hu Funding details: Hungarian Scientific Research Fund, OTKA, OTKA K113150 Funding text 1: This project was supported by the Hungarian Scientific Research Fund (OTKA K113150). Department of Organic Chemistry and Technology, Budapest University of Technology and Economics, Gellért tér 4, Budapest, H-1111, Hungary Quality Process Development Department, Egis Pharmaceuticals Plc, Keresztúri út 30-38, Budapest, H-1106, Hungary Spectroscopic Research Department, Gedeon Richter Plc, 10, P. O. Box 27, Budapest, H-1475, Hungary Department of Organic Chemistry, University of Szeged, Dóm tér 8, Szeged, H-6720, Hungary Cited By :1 Export Date: 26 May 2021 CODEN: CORCF Correspondence Address: Keglevich, P.; Department of Organic Chemistry and Technology, Gellért tér 4, Hungary; email: pkeglevich@mail.bme.hu Funding details: Hungarian Scientific Research Fund, OTKA, OTKA K113150 Funding text 1: This project was supported by the Hungarian Scientific Research Fund (OTKA K113150). Department of Organic Chemistry and Technology, Budapest University of Technology and Economics, Gellért tér 4, Budapest, H-1111, Hungary Quality Process Development Department, Egis Pharmaceuticals Plc, Keresztúri út 30-38, Budapest, H-1106, Hungary Spectroscopic Research Department, Gedeon Richter Plc, 10, P. O. Box 27, Budapest, H-1475, Hungary Department of Organic Chemistry, University of Szeged, Dóm tér 8, Szeged, H-6720, Hungary Cited By :1 Export Date: 4 June 2021 CODEN: CORCF Correspondence Address: Keglevich, P.; Department of Organic Chemistry and Technology, Gellért tér 4, Hungary; email: pkeglevich@mail.bme.hu Funding details: Hungarian Scientific Research Fund, OTKA, OTKA K113150 Funding text 1: This project was supported by the Hungarian Scientific Research Fund (OTKA K113150). Funding Agency and Grant Number: Hungarian Scientific Research FundOrszagos Tudomanyos Kutatasi Alapprogramok (OTKA) [OTKA K113150] Funding text: This project was supported by the Hungarian Scientific Research Fund (OTKA K113150). Department of Organic Chemistry and Technology, Budapest University of Technology and Economics, Gellért tér 4, Budapest, H-1111, Hungary Quality Process Development Department, Egis Pharmaceuticals Plc, Keresztúri út 30-38, Budapest, H-1106, Hungary Spectroscopic Research Department, Gedeon Richter Plc, 10, P. O. Box 27, Budapest, H-1475, Hungary Department of Organic Chemistry, University of Szeged, Dóm tér 8, Szeged, H-6720, Hungary Cited By :2 Export Date: 13 July 2021 CODEN: CORCF Correspondence Address: Keglevich, P.; Department of Organic Chemistry and Technology, Gellért tér 4, Hungary; email: pkeglevich@mail.bme.hu Funding details: Hungarian Scientific Research Fund, OTKA, OTKA K113150 Funding text 1: This project was supported by the Hungarian Scientific Research Fund (OTKA K113150). LA - English DB - MTMT ER - TY - JOUR AU - Herman, Bianka Edina AU - Kiss, Anita AU - Wölfling, János AU - Mernyák, Erzsébet AU - Szécsi, Mihály AU - Schneider, Gyula TI - Synthesis of substituted 15β-alkoxy estrone derivatives and their cofactor-dependent inhibitory effect on 17β-HSD1 JF - JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY J2 - J ENZYM INHIB MED CH VL - 34 PY - 2019 IS - 1 SP - 1271 EP - 1286 PG - 16 SN - 1475-6366 DO - 10.1080/14756366.2019.1634064 UR - https://m2.mtmt.hu/api/publication/30747981 ID - 30747981 N1 - Export Date: 6 August 2019 LA - English DB - MTMT ER - TY - JOUR AU - Kiss, Anita AU - Wölfling, János AU - Mernyák, Erzsébet AU - Nagyné Frank, Éva AU - Gyovai, András AU - Kulmány, Ágnes Erika AU - Zupkó, István AU - Schneider, Gyula TI - Stereoselective Synthesis of New Type of Estradiol Hybrid Molecules and their Antiproliferative Activities JF - STEROIDS J2 - STEROIDS VL - 148 PY - 2019 SP - 63 EP - 72 PG - 10 SN - 0039-128X DO - 10.1016/j.steroids.2019.02.016 UR - https://m2.mtmt.hu/api/publication/30672538 ID - 30672538 LA - English DB - MTMT ER - TY - JOUR AU - Angyal, Anikó AU - András, Demjén AU - Harmat, Veronika AU - Wölfling, János AU - László, G. Puskás AU - Kanizsai, Iván TI - 1,3-Dipolar Cycloaddition of Isatin-Derived Azomethine Ylides with 2H-Azirines: Stereoselective Synthesis of 1,3-Diazaspiro[bicyclo[3.1.0]hexane]oxindoles JF - JOURNAL OF ORGANIC CHEMISTRY J2 - J ORG CHEM VL - 84 PY - 2019 IS - 7 SP - 4273 EP - 4281 PG - 9 SN - 0022-3263 DO - 10.1021/acs.joc.9b00242 UR - https://m2.mtmt.hu/api/publication/30641393 ID - 30641393 N1 - AVIDIN Ltd., Alsó kiköto sor 11/D, Szeged, H-6726, Hungary Department of Organic Chemistry, University of Szeged, Dóm tér 8, Szeged, H-6720, Hungary Laboratory of Structural Chemistry and Biology, MTA-ELTE Protein Modeling Research Group, Institute of Chemistry, Eötvös Loránd University, Pázmány P. sétány 1/A, Budapest, H-1117, Hungary Cited By :16 Export Date: 27 January 2022 CODEN: JOCEA Correspondence Address: Kanizsai, I.; AVIDIN Ltd., Alsó kiköto sor 11/D, Hungary; email: i.kanizsai@avidinbiotech.com LA - English DB - MTMT ER - TY - JOUR AU - Jopp, Stefan AU - Ehlers, Peter AU - Nagyné Frank, Éva AU - Mernyák, Erzsébet AU - Schneider, Gyula AU - Wölfling, János AU - Villinger, Alexander AU - Langer, Peter TI - Site-Selective Synthesis of 3,17-Diaryl-1,3,5,16-estratetraenes JF - SYNLETT J2 - SYNLETT VL - 30 ET - 0 PY - 2019 IS - 5 SP - 600 EP - 604 PG - 5 SN - 0936-5214 DO - 10.1055/s-0037-1611720 UR - https://m2.mtmt.hu/api/publication/30429176 ID - 30429176 LA - English DB - MTMT ER -