1.
Garami, Kristóf ; Péczka, Nikolett ; Petri, László ; Imre, Tímea ; Langó, Tamás ; Szabó, Zoltán ; Orgován, Zoltán ; Szabó, Pál ; Keserű, György Miklós ✉ ; Ábrányi-Balogh, Péter ✉
Target agnostic photoaffinity labelling by sulfonylhydrazones
ANGEWANDTE CHEMIE-INTERNATIONAL EDITION 64 : 17 Paper: e202408701 , 7 p. (2025)
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Publication:35781560 Validated Core Citing Journal Article (Article ) Scientific
Article (Journal Article) | Scientific[35781560] [Validated]
2.
Wéber, Edit ; Ábrányi-Balogh, Péter* ; Martinek, Tamas A. ; Nagymihály, Bence ; Menyhárd, Dóra Karancsiné ; Péczka, Nikolett ; Gadanecz, Márton ; Schlosser, Gitta ; Orgován, Zoltán ; Bogár, Ferenc et al.
Target‐templated Construction of Functional Proteomimetics Using Photo‐foldamer Libraries
ANGEWANDTE CHEMIE 137 : 2 Paper: e202410435 (2025)
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Locked Publication:35427664 Published Core Journal Article (Republication ) Scientific
Republication (Journal Article) | Scientific[35427664] [Approved]
3.
Ábrányi-Balogh, Péter ; Bajusz, Dávid* ; Orgován, Zoltán* ; Keeley, Aaron B. ; Petri, László ; Péczka, Nikolett ; Szalai, Tibor Viktor ; Pálfy, Gyula ; Gadanecz, Márton ; Grant, Emma K. et al.
Mapping protein binding sites by photoreactive fragment pharmacophores
COMMUNICATIONS CHEMISTRY 7 : 1 Paper: 168 , 13 p. (2024)
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Locked Publication:35160281 Validated Core Citing Journal Article (Article ) Scientific
Article (Journal Article) | Scientific[35160281] [Validated]
4.
Keeley, Aaron B. ; Kopranovic, Aleksandra ; Di Lorenzo, Vincenzo ; Ábrányi-Balogh, Péter ; Jänsch, Niklas ; Lai, Linh N. ; Petri, László ; Orgován, Zoltán ; Pölöske, Daniel ; Orlova, Anna et al.
Electrophilic MiniFrags Revealed Unprecedented Binding Sites for Covalent HDAC8 Inhibitors
JOURNAL OF MEDICINAL CHEMISTRY 67 : 1 pp. 572-585. , 14 p. (2024)
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Locked Publication:34445373 Validated Core Citing Journal Article (Article ) Scientific
Citing papers: 6 | Independent citation: 5 | Self citation: 1 | Unknown citation: 0 | Number of citations in WoS: 6 | Number of citations in Scopus: 3 | WoS/Scopus assigned: 6 | Number of citations with DOI: 6
Article (Journal Article) | Scientific[34445373] [Validated]
All citations+mentions: 6, External citations: 5, Self citations: 1, Unhandled citations: 0
5.
Péczka, Nikolett ; Ranđelović, Ivan ; Orgován, Zoltán ; Csorba, Noémi ; Egyed, Attila ; Petri, László ; Ábrányi-Balogh, Péter ; Gadanecz, Márton ; Perczel, András ; Tóvári, József et al.
Contribution of Noncovalent Recognition and Reactivity to the Optimization of Covalent Inhibitors : A Case Study on KRasG12C
ACS CHEMICAL BIOLOGY 19 : 8 pp. 1743-1756. , 14 p. (2024)
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Locked Publication:35134356 Validated Core Citing Journal Article (Article ) Scientific
Citing papers: 1 | Independent citation: 1 | Self citation: 0 | Unknown citation: 0 | Number of citations in WoS: 1 | Number of citations in Scopus: 1 | WoS/Scopus assigned: 1 | Number of citations with DOI: 1
Article (Journal Article) | Scientific[35134356] [Validated]
All citations+mentions: 1, External citations: 1, Self citations: 0, Unhandled citations: 0
6.
Orgován, Zoltán
Computational investigation of the allosteric modulation of metabotropic glutamate receptor 5 163 p.
Budapest University of Technology and Economics, Budapesti Műszaki és Gazdaságtudományi Egyetem, Oláh György Doktori Iskola, Keserű György Miklós Accepted: 2023 Published/defended: 2023
Műegyetem Digitális Archívum ODT védés
Publication:34738155 Published Core Thesis (PhD ) Scientific
PhD (Thesis) | Scientific[34738155] [Approved]
7.
Orgován, Zoltán ; Péczka, Nikolett* ; Petri, László ; Ábrányi-Balogh, Péter ; Ranđelović, Ivan ; Tóth, Szilárd ; Szakács, Gergely ; Nyíri, Kinga ; Vértessy, Beáta ; Pálfy, Gyula et al.
Covalent fragment mapping of KRasG12C revealed novel chemotypes with in vivo potency
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY 250 Paper: 115212 , 7 p. (2023)
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Locked Publication:33647485 Admin approved Core Citing Journal Article (Article ) Scientific
Citing papers: 3 | Independent citation: 1 | Self citation: 2 | Unknown citation: 0 | Number of citations in WoS: 2 | Number of citations in Scopus: 3 | WoS/Scopus assigned: 3 | Number of citations with DOI: 3
Article (Journal Article) | Scientific[33647485] [Admin approved]
All citations+mentions: 3, External citations: 1, Self citations: 2, Unhandled citations: 0
8.
Kiss-Szemán, Anna J. ; Takács, Luca ; Orgován, Zoltán ; Stráner, Pál ; Jákli, Imre ; Schlosser, Gitta ; Masiulis, Simonas ; Harmat, Veronika ; Menyhárd, Dóra K. ; Perczel, András
A carbapenem antibiotic inhibiting a mammalian serine protease: structure of the acylaminoacyl peptidase–meropenem complex
CHEMICAL SCIENCE 13 : 48 pp. 14264-14276. , 13 p. (2022)
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Publication:33307131 Validated Core Citing Journal Article (Article ) Scientific
Citing papers: 3 | Independent citation: 3 | Self citation: 0 | Unknown citation: 0 | Number of citations in WoS: 3 | Number of citations in Scopus: 3 | WoS/Scopus assigned: 3 | Number of citations with DOI: 3
Article (Journal Article) | Scientific[33307131] [Validated]
All citations+mentions: 3, External citations: 3, Self citations: 0, Unhandled citations: 0
9.
Peczka, Nikolett ; Orgovan, Zoltan ; Abranyi-Balogh, Peter ; Keseru, Gyorgy Miklos ✉
Electrophilic warheads in covalent drug discovery: an overview
EXPERT OPINION ON DRUG DISCOVERY 17 : 4 pp. 413-422. , 10 p. (2022)
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Locked Publication:32756662 Admin approved Core Citing Journal Article (Survey paper ) Scientific
Citing papers: 40 | Independent citation: 37 | Self citation: 3 | Unknown citation: 0 | Number of citations in WoS: 40 | Number of citations in Scopus: 18 | WoS/Scopus assigned: 40 | Number of citations with DOI: 40
Survey paper (Journal Article) | Scientific[32756662] [Admin approved]
All citations+mentions: 40, External citations: 37, Self citations: 3, Unhandled citations: 0
10.
Orgovan, Zoltan ; Ferenczy, Gyorgy G. ; Keseru, Gyorgy M. ✉
Allosteric Molecular Switches in Metabotropic Glutamate Receptors
CHEMMEDCHEM 16 : 1 pp. 81-93. , 14 p. (2021)
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Citing papers: 12 | Independent citation: 12 | Self citation: 0 | Unknown citation: 0 | Number of citations in WoS: 12 | Number of citations in Scopus: 6 | WoS/Scopus assigned: 12 | Number of citations with DOI: 12
Survey paper (Journal Article) | Scientific[31698584] [Validated]
All citations+mentions: 12, External citations: 12, Self citations: 0, Unhandled citations: 0
11.
Jójárt, Balázs ; Orgován, Zoltán* ; Márki, Árpád ; Pándy-Szekeres, Gáspár ; Ferenczy, György G. ; Keserű, György M. ✉
Allosteric activation of metabotropic glutamate receptor 5
JOURNAL OF BIOMOLECULAR STRUCTURE & DYNAMICS 38 : 9 pp. 2624-2632. , 10 p. (2020)
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Locked Publication:30834454 Validated Core Citing Journal Article (Article ) Scientific
Citing papers: 5 | Independent citation: 3 | Self citation: 2 | Unknown citation: 0 | Number of citations in WoS: 5 | Number of citations in Scopus: 5 | WoS/Scopus assigned: 5 | Number of citations with DOI: 5
Article (Journal Article) | Scientific[30834454] [Validated]
All citations+mentions: 5, External citations: 3, Self citations: 2, Unhandled citations: 0
12.
Menyhard, Dora K. ; Palfy, Gyula ; Orgovan, Zoltan ; Vida, Istvan ; Keseru, Gyorgy M. ✉ ; Perczel, Andras ✉
Structural impact of GTP binding on downstream KRAS signaling
CHEMICAL SCIENCE 11 : 34 pp. 9272-9289. , 18 p. (2020)
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Locked Publication:31605838 Validated Core Citing Journal Article (Article ) Scientific
Citing papers: 34 | Independent citation: 31 | Self citation: 3 | Unknown citation: 0 | Number of citations in WoS: 29 | Number of citations in Scopus: 31 | WoS/Scopus assigned: 31 | Number of citations with DOI: 32
Article (Journal Article) | Scientific[31605838] [Validated]
All citations+mentions: 34, External citations: 31, Self citations: 3, Unhandled citations: 0
13.
Orgován, Z. ; Keserű, G.M. ✉
Small molecule inhibitors of RAS proteins with oncogenic mutations
CANCER AND METASTASIS REVIEWS 39 : 4 pp. 1107-1126. , 20 p. (2020)
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Locked Publication:31473660 Admin approved Core Citing Journal Article (Survey paper ) Scientific
Citing papers: 19 | Independent citation: 15 | Self citation: 4 | Unknown citation: 0 | Number of citations in WoS: 19 | Number of citations in Scopus: 13 | WoS/Scopus assigned: 19 | Number of citations with DOI: 19
Survey paper (Journal Article) | Scientific[31473660] [Admin approved]
All citations+mentions: 19, External citations: 15, Self citations: 4, Unhandled citations: 0
14.
Szabó, György ; Kolok, Sándor ; Orgován, Zoltán ; Vastag, Mónika ; Béni, Zoltán ; Kóti, János ; Sághy, Katalin ; Lévay, György I. ; Greiner, István ; Keserű, György M. ✉
Discovery of dihydropyrazino-benzimidazole derivatives as metabotropic glutamate receptor-2 (mGluR2) positive allosteric modulators (PAMs)
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY 186 Paper: 111881 , 17 p. (2020)
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Article (Journal Article) | Scientific[30928052] [Validated]
All citations+mentions: 5, External citations: 4, Self citations: 1, Unhandled citations: 0
15.
Christopher, John A. ✉ ; Orgován, Zoltán ; Congreve, Miles ; Doré, Andrew S. ; Errey, James C. ; Marshall, Fiona H. ; Mason, Jonathan S. ; Okrasa, Krzysztof ; Rucktooa, Prakash ; Serrano-Vega, Maria J. et al.
Structure-Based Optimization Strategies for G Protein-Coupled Receptor (GPCR) Allosteric Modulators: A Case Study from Analyses of New Metabotropic Glutamate Receptor 5 (mGlu 5 ) X-ray Structures
JOURNAL OF MEDICINAL CHEMISTRY 62 : 1 pp. 207-222. , 16 p. (2019)
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Locked Publication:30334026 Validated Core Citing Journal Article (Article ) Scientific
Citing papers: 60 | Independent citation: 52 | Self citation: 8 | Unknown citation: 0 | Number of citations in WoS: 60 | Number of citations in Scopus: 42 | WoS/Scopus assigned: 60 | Number of citations with DOI: 60
Article (Journal Article) | Scientific[30334026] [Validated]
All citations+mentions: 60, External citations: 52, Self citations: 8, Unhandled citations: 0
16.
Nyíri, Kinga ; Koppány, Gergely ; Pálfy, Gyula ; Vida, István ; Tóth, Szilárd ; Orgován, Zoltán ; Ivan, Ranđelović ; Baranyi, Marcell ; Molnár, Eszter ; Keserű, György Miklós et al.
Allélspecifikus inhibitorok nyomában: a RASopátia konzorcium célpontjában a KRAS fehérje onkogén mutációi
MAGYAR ONKOLÓGIA 63 : 4 pp. 310-323. , 10 p. (2019)
Scopus PubMed Other URL Matarka MOB
Locked Publication:31038395 Validated Core Citing Journal Article (Article ) Scientific
Article (Journal Article) | Scientific[31038395] [Validated]
17.
Orgován, Zoltán ; Ferenczy, György G. ; Keserű, György M. ✉
Fragment-Based Approaches for Allosteric Metabotropic Glutamate Receptor (mGluR) Modulators
CURRENT TOPICS IN MEDICINAL CHEMISTRY 19 : 19 pp. 1768-1781. , 14 p. (2019)
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Citing papers: 7 | Independent citation: 5 | Self citation: 2 | Unknown citation: 0 | Number of citations in WoS: 7 | Number of citations in Scopus: 3 | WoS/Scopus assigned: 7 | Number of citations with DOI: 7
Survey paper (Journal Article) | Scientific[30834430] [Validated]
All citations+mentions: 7, External citations: 5, Self citations: 2, Unhandled citations: 0
18.
Orgován, Zoltán ; Ferenczy, György G. ; Keserű, György M. ✉
The role of water and protein flexibility in the structure-based virtual screening of allosteric GPCR modulators: an mGlu5 receptor case study
JOURNAL OF COMPUTER-AIDED MOLECULAR DESIGN 33 : 9 pp. 787-797. , 11 p. (2019)
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Locked Publication:30834424 Validated Core Citing Journal Article (Article ) Scientific
Citing papers: 6 | Independent citation: 6 | Self citation: 0 | Unknown citation: 0 | Number of citations in WoS: 6 | Number of citations in Scopus: 3 | WoS/Scopus assigned: 6 | Number of citations with DOI: 6
Article (Journal Article) | Scientific[30834424] [Validated]
All citations+mentions: 6, External citations: 6, Self citations: 0, Unhandled citations: 0
19.
Orgován, Zoltán ; Ferenczy, György G ; Steinbrecher, Thomas ; Szilágyi, Bence ; Bajusz, Dávid ; Keserű, György M ✉
Validation of tautomeric and protomeric binding modes by free energy calculations. A case study for the structure based optimization of d-amino acid oxidase inhibitors
JOURNAL OF COMPUTER-AIDED MOLECULAR DESIGN 32 : 2 pp. 331-345. , 15 p. (2018)
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Locked Publication:3333356 Validated Core Citing Journal Article (Article ) Scientific
Citing papers: 8 | Independent citation: 5 | Self citation: 3 | Unknown citation: 0 | Number of citations in WoS: 8 | Number of citations in Scopus: 5 | WoS/Scopus assigned: 8 | Number of citations with DOI: 8
Article (Journal Article) | Scientific[3333356] [Validated]
All citations+mentions: 8, External citations: 5, Self citations: 3, Unhandled citations: 0
20.
Galambos, J ; Bielik, A ; Wágner, G ; Domány, G ; Kóti, J ; Béni, Z ; Szigetvári, Á ; Sánta, Z ; Orgován, Z ; Bobok, A et al.
Discovery of 4-amino-3-arylsulfoquinolines, a novel non-acetylenic chemotype of metabotropic glutamate 5 (mGlu5) receptor negative allosteric modulators
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY 133 pp. 240-254. , 15 p. (2017)
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Locked Publication:3291826 Validated Core Journal Article (Article ) Scientific
Citing papers: 8 | Independent citation: 6 | Self citation: 2 | Unknown citation: 0 | Number of citations in WoS: 8 | Number of citations in Scopus: 8 | WoS/Scopus assigned: 8 | Number of citations with DOI: 8
Article (Journal Article) | Scientific[3291826] [Validated]
All citations+mentions: 8, External citations: 6, Self citations: 2, Unhandled citations: 0
2025-05-20 09:12