1.
Szilágyi, Bence ; Egyed, Attila ; Mándity, István ; Nagy, Tamás ; Kátai-Fadgyas, Katalin ; Volk, Balázs ✉ ; Keserű György, M.
Safe and Efficient Continuous-Flow Synthesis and Batchwise Hydrolysis of Ethyl 5-Acetyl-1H-pyrazole-3-carboxylate: A Key Synthon of Darolutamide
SYNTHESIS-STUTTGART 55 : 6 pp. 959-966. , 8 p. (2023)
DOI WoS Scopus
Publication:33283298 Admin approved Core Journal Article (Study Group ) Scientific
Study Group (Journal Article) | Scientific[33283298] [Admin approved]
2.
Poszávácz, László ; Szilágyi, Bence ; Nagy, Tamás ; Egyed, Attila ; Kátai-Fadgyas, Katalin ; Keserű, György M. ; Mándity, István ; Volk, Balázs
„Semmi sem olyan egyszerű, mint amilyennek látszik”. Darolutamid intermedier generikus szemmel (2022)
Előadás, Gyógyszerkémiai és Gyógyszertechnológiai Szimpózium '22, Herceghalom (2022. szeptember 19-20.),
Publication:33106229 Admin approved Core Miscellaneous (Not classified ) Scientific
Not classified (Miscellaneous) | Scientific[33106229] [Admin approved]
3.
Kollár, Levente ; Gobec, Martina* ; Szilágyi, Bence ; Proj, Matic ; Knez, Damijan ; Ábrányi-Balogh, Péter ; Petri, László ; Imre, Tímea ; Bajusz, Dávid ; Ferenczy, György G. et al.
Discovery of selective fragment-sized immunoproteasome inhibitors
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY 219 Paper: 113455 , 23 p. (2021)
DOI REAL WoS Scopus PubMed
Publication:31984014 Validated Core Citing Journal Article (Article ) Scientific
Citing papers: 5 | Independent citation: 1 | Self citation: 4 | Unknown citation: 0 | Number of citations in WoS: 4 | Number of citations in Scopus: 4 | WoS/Scopus assigned: 5 | Number of citations with DOI: 5
Article (Journal Article) | Scientific[31984014] [Validated]
All citations+mentions: 5, External citations: 1, Self citations: 4, Unhandled citations: 0
4.
Szepesi Kovács, Dénes ; Hajdu, Imre ; Mészáros, Gergely ; Wittner, Lucia ; Meszéna, Domokos ; Tóth, Estilla Zsófia ; Hegedűs, Zita ; Ranđelović, Ivan ; Tóvári, József ; Szabó, Tímea et al.
Synthesis and characterization of new fluorescent boro-β-carboline dyes
RSC ADVANCES 11 : 21 pp. 12802-12807. , 6 p. (2021)
DOI WoS Scopus
Locked Publication:31951354 Validated Core Citing Journal Article (Article ) Scientific
Citing papers: 3 | Independent citation: 3 | Self citation: 0 | Unknown citation: 0 | Number of citations in WoS: 3 | Number of citations in Scopus: 3 | WoS/Scopus assigned: 3 | Number of citations with DOI: 3
Article (Journal Article) | Scientific[31951354] [Validated]
All citations+mentions: 3, External citations: 3, Self citations: 0, Unhandled citations: 0
5.
Szilágyi, Bence
Design and synthesis of D-amino acid oxidase inhibitors
Budapesti Műszaki és Gazdaságtudományi Egyetem, Oláh György Doktori Iskola, Keserű György Miklós Published/defended: 2019
Teljes dokumentum
Publication:31353710 Admin approved Core Thesis (PhD ) Scientific
PhD (Thesis) | Scientific[31353710] [Admin approved]
6.
Szilágyi, Bence ; Hargitai, Csilla ; Kelemen, Ádám A. ; Rácz, Anita ; Ferenczy, György G. ; Volk, Balázs ✉ ; Keserű, György M. ✉
Synthesis and Biochemical Evaluation of Lid-Open D-Amino Acid Oxidase Inhibitors
MOLECULES 24 : 2 Paper: 290 , 8 p. (2019)
DOI WoS Scopus PubMed Egyéb URL
Publication:30392129 Validated Core Journal Article (Article ) Scientific
Article (Journal Article) | Scientific[30392129] [Validated]
7.
Orgován, Zoltán ; Ferenczy, György G ; Steinbrecher, Thomas ; Szilágyi, Bence ; Bajusz, Dávid ; Keserű, György M ✉
Validation of tautomeric and protomeric binding modes by free energy calculations. A case study for the structure based optimization of d-amino acid oxidase inhibitors
JOURNAL OF COMPUTER-AIDED MOLECULAR DESIGN 32 : 2 pp. 331-345. , 15 p. (2018)
DOI WoS Scopus PubMed
Publication:3333356 Validated Core Citing Journal Article (Article ) Scientific
Citing papers: 7 | Independent citation: 4 | Self citation: 3 | Unknown citation: 0 | Number of citations in WoS: 7 | Number of citations in Scopus: 5 | WoS/Scopus assigned: 7 | Number of citations with DOI: 7
Article (Journal Article) | Scientific[3333356] [Validated]
All citations+mentions: 7, External citations: 4, Self citations: 3, Unhandled citations: 0
8.
Szilágyi, B ; Skok, Ž ; Rácz, A ; Frlan, R ; Ferenczy, GG ; Ilaš, J ; Keserű, GM ✉
Discovery of D-amino acid oxidase inhibitors based on virtual screening against the lid-open enzyme conformation
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS 28 : 10 pp. 1693-1698. , 6 p. (2018)
DOI WoS Scopus PubMed
Publication:3375019 Validated Core Citing Journal Article (Article ) Scientific
Citing papers: 5 | Independent citation: 5 | Self citation: 0 | Unknown citation: 0 | Number of citations in WoS: 4 | Number of citations in Scopus: 2 | WoS/Scopus assigned: 4 | Number of citations with DOI: 4
Article (Journal Article) | Scientific[3375019] [Validated]
All citations+mentions: 5, External citations: 5, Self citations: 0, Unhandled citations: 0
9.
Szilágyi, B. ; Ferenczy, G.G. ; Keserű, G.M. ✉
Drug discovery strategies and the preclinical development of D-amino-acid oxidase inhibitors as antipsychotic therapies
EXPERT OPINION ON DRUG DISCOVERY 13 : 10 pp. 973-982. , 10 p. (2018)
DOI WoS Scopus PubMed
Publication:30353690 Validated Core Citing Journal Article (Survey paper ) Scientific
Citing papers: 6 | Independent citation: 5 | Self citation: 1 | Unknown citation: 0 | Number of citations in WoS: 6 | Number of citations in Scopus: 5 | WoS/Scopus assigned: 6 | Number of citations with DOI: 6
Survey paper (Journal Article) | Scientific[30353690] [Validated]
All citations+mentions: 6, External citations: 5, Self citations: 1, Unhandled citations: 0
10.
Szilagyi, B ; Kovacs, P ; Ferenczy, GG ; Racz, A ; Nemeth, K ; Visy, J ; Szabo, P ; Ilas, J ; Balogh, GT ; Monostory, K et al.
Discovery of isatin and 1H-indazol-3-ol derivatives as d-amino acid oxidase (DAAO) inhibitors
BIOORGANIC & MEDICINAL CHEMISTRY 26 : 8 pp. 1579-1587. , 9 p. (2018)
DOI SE Repozitórium WoS Scopus PubMed Google scholar
Locked Publication:3344151 Admin approved Core Citing Journal Article (Article ) Scientific
Citing papers: 8 | Independent citation: 7 | Self citation: 1 | Unknown citation: 0 | Number of citations in WoS: 8 | Number of citations in Scopus: 8 | WoS/Scopus assigned: 8 | Number of citations with DOI: 8
Article (Journal Article) | Scientific[3344151] [Admin approved]
All citations+mentions: 8, External citations: 7, Self citations: 1, Unhandled citations: 0
11.
L, Somsák ; M, Polyák ; G, Varga ; J, Begum ; B, Szilágyi ; L, Juhász ; T, Docsa ; P, Gergely ; J M, Hayes
N-(β-D-Glucopyranosyl) Oxadiazole- and 1,2,4-Triazolecarboxamides as Glycogen Phosphorylase Inhibitors: Synthesis, Enzyme Kinetics and Computational Evaluation
In: 27th International Carbohydrate Symposium
Bengaluru, India : Indian Institute of Science, (2014) Paper: I-P-58
Publication:2517810 Admin approved Core Conference paper (Abstract )
Abstract (Conference paper) | Scientific[2517810] [Admin approved]
12.
Mária, Polyák ; Gergő, Varga ; Bence, Szilágyi ; Tibor, Docsa ; Pál, Gergely ; László, Juhász ; László, Somsák
Synthesis and enzyme kinetic evaluation of heterocyclic bioisosteric analogues of N-acyl-N’-β-D-glucopyranosyl urea type glycogen phosphorylase inhibitors
In: Ernest, Giralt (eds.) 5th European Conference on Chemistry for Life Sciences, Abstract Book
Barcelona, Spain (2013) p. 93
Publication:2382460 Admin approved Core Conference paper (Abstract )
Abstract (Conference paper) | Scientific[2382460] [Admin approved]
13.
Polyák, M ; Varga, G ; Szilágyi, B ; Juhász, L ; Docsa, T ; Gergely, P ; Begum, J ; Hayes, JM ; Somsák, L ✉
Synthesis, enzyme kinetics and computational evaluation of N-(beta-D-glucopyranosyl) oxadiazolecarboxamides as glycogen phosphorylase inhibitors
BIOORGANIC & MEDICINAL CHEMISTRY 21 pp. 5738-5747. , 10 p. (2013)
DOI REAL WoS DEA Scopus PubMed Teljes dokumentum
Publication:2381496 Published Core Citing Journal Article (Article ) Scientific
Citing papers: 20 | Independent citation: 10 | Self citation: 10 | Unknown citation: 0 | Number of citations in WoS: 15 | Number of citations in Scopus: 12 | WoS/Scopus assigned: 16 | Number of citations with DOI: 16
Article (Journal Article) | Scientific[2381496] [Approved]
All citations+mentions: 20, External citations: 10, Self citations: 10, Unhandled citations: 0
14.
Polyák, Mária ; Varga, Gergely ; Szilágyi, Bence ; Docsa, Tibor ; Gergely, Pál ; Juhász, László ; Somsák, László
N-Acil-N’-β-D-glükopiranozil-karbamid típusú glikogén foszforiláz inhibitorok heterociklusos bioizosztér analógjainak szintézise és enzimkinetikai vizsgálata
In: Magyar, Kémikusok Egyesülete (eds.) Vegyészkonferencia 2013 : 2013. június 26-28., Hajdúszoboszló : program és elődásösszefoglalók
Bp, Hungary : Magyar Kémikusok Egyesülete (MKE) (2013) 152 p. p. 114 Paper: P-54
Publication:2382468 Admin approved Core Chapter in Book (Abstract ) Scientific
Abstract (Chapter in Book) | Scientific[2382468] [Admin approved]
15.
Marietta, Tóth ; Gergely, Tibor Varga ; Mária, Polyák ; Bence, Szilágyi ; Sándor, Kun ; I, Takács ; László, Juhász ; Tibor, Docsa ; Pál, Gergely ; László, Somsák
SAR study of glycogen phosphorylase inhibitors: heterocycles as bioisosteric amide replacements in N-acyl-beta-D-glucopyranosylamines and N-acyl-N’-beta-D-glucopyranosyl ureas
In: 26th International Carbohydrate Symposium
(2012) Paper: P122
Publication:2314255 Admin approved Core Conference paper (Abstract )
Abstract (Conference paper) | Scientific[2314255] [Admin approved]
16.
Tóth, M ; Varga, G T ; Polyák, M ; Szilágyi, B ; Kun, S ; Takács, I ; Juhász, L ; Docsa, T ; Gergely, P ; Somsák, L
SAR Study of Glycogen Phosphorylase Inhibitors: Heterocycles as Bioisosteric Amide Replacements in N-Acyl-beta-D-Glucopyranosylamines and N-Acyl-N’-beta-D-Glucopyranosyl Ureas
In: 26th International Carbohydrate Symposium
(2012) pp. F80-F80.
Publication:2034044 Admin approved Core Conference paper (Abstract )
Abstract (Conference paper) | Scientific[2034044] [Admin approved]
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