MTMT2: publication list

Szilágyi, Bence ; Egyed, Attila ; Mándity, István ; Nagy, Tamás ; Kátai-Fadgyas, Katalin ; Volk, Balázs ✉ ; Keserű György, M. ✉

Safe and Efficient Continuous-Flow Synthesis and Batchwise Hydrolysis of Ethyl 5-Acetyl-1H-pyrazole-3-carboxylate: A Key Synthon of Darolutamide

SYNTHESIS-STUTTGART 55 : 6 pp. 959-966. , 8 p. (2023)

DOI WoS Scopus

Locked Publication:33283298 Validated Core Journal Article (Article ) Scientific

Article (Journal Article) | Scientific[33283298] [Validated]

All citations+mentions: 1, External citations: 0, Self citations: 1, Unhandled citations: 0

Poszávácz, László ; Szilágyi, Bence ; Nagy, Tamás ; Egyed, Attila ; Kátai-Fadgyas, Katalin ; Keserű, György M. ; Mándity, István ; Volk, Balázs

„Semmi sem olyan egyszerű, mint amilyennek látszik”. Darolutamid intermedier generikus szemmel (2022)

Előadás, Gyógyszerkémiai és Gyógyszertechnológiai Szimpózium '22, Herceghalom (2022. szeptember 19-20.),

Publication:33106229 Admin approved Core Miscellaneous (Not classified ) Scientific

Not classified (Miscellaneous) | Scientific[33106229] [Admin approved]

Kollár, Levente ; Gobec, Martina^* ; Szilágyi, Bence ; Proj, Matic ; Knez, Damijan ; Ábrányi-Balogh, Péter ; Petri, László ; Imre, Tímea ; Bajusz, Dávid ; Ferenczy, György G. et al.

Discovery of selective fragment-sized immunoproteasome inhibitors

EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY 219 Paper: 113455 , 23 p. (2021)

DOI REAL WoS Scopus PubMed

Publication:31984014 Validated Core Citing Journal Article (Article ) Scientific

Article (Journal Article) | Scientific[31984014] [Validated]

All citations+mentions: 11, External citations: 6, Self citations: 5, Unhandled citations: 0

Szepesi Kovács, Dénes ; Hajdu, Imre ; Mészáros, Gergely ; Wittner, Lucia ; Meszéna, Domokos ; Tóth, Estilla Zsófia ; Hegedűs, Zita ; Ranđelović, Ivan ; Tóvári, József ; Szabó, Tímea et al.

Synthesis and characterization of new fluorescent boro-β-carboline dyes

RSC ADVANCES 11 : 21 pp. 12802-12807. , 6 p. (2021)

DOI WoS Scopus PubMed Google scholar

Locked Publication:31951354 Validated Core Citing Journal Article (Article ) Scientific

Article (Journal Article) | Scientific[31951354] [Validated]

All citations+mentions: 12, External citations: 9, Self citations: 3, Unhandled citations: 0

Szilágyi, Bence

Design and synthesis of D-amino acid oxidase inhibitors

Budapest University of Technology and Economics, Oláh György Doktori Iskola, Keserű György Miklós Published/defended: 2019

Teljes dokumentum

Publication:31353710 Admin approved Core Thesis (PhD ) Scientific

PhD (Thesis) | Scientific[31353710] [Admin approved]

Szilágyi, Bence ; Hargitai, Csilla ; Kelemen, Ádám A. ; Rácz, Anita ; Ferenczy, György G. ; Volk, Balázs ✉ ; Keserű, György M. ✉

Synthesis and Biochemical Evaluation of Lid-Open D-Amino Acid Oxidase Inhibitors

MOLECULES 24 : 2 Paper: 290 , 8 p. (2019)

DOI WoS Scopus PubMed Other URL

Publication:30392129 Validated Core Journal Article (Article ) Scientific

Article (Journal Article) | Scientific[30392129] [Validated]

All citations+mentions: 1, External citations: 1, Self citations: 0, Unhandled citations: 0

Orgován, Zoltán ; Ferenczy, György G ; Steinbrecher, Thomas ; Szilágyi, Bence ; Bajusz, Dávid ; Keserű, György M ✉

Validation of tautomeric and protomeric binding modes by free energy calculations. A case study for the structure based optimization of d-amino acid oxidase inhibitors

JOURNAL OF COMPUTER-AIDED MOLECULAR DESIGN 32 : 2 pp. 331-345. , 15 p. (2018)

DOI WoS Scopus PubMed

Publication:3333356 Validated Core Citing Journal Article (Article ) Scientific

Article (Journal Article) | Scientific[3333356] [Validated]

All citations+mentions: 8, External citations: 5, Self citations: 3, Unhandled citations: 0

Szilágyi, B ; Skok, Ž ; Rácz, A ; Frlan, R ; Ferenczy, GG ; Ilaš, J ; Keserű, GM ✉

Discovery of D-amino acid oxidase inhibitors based on virtual screening against the lid-open enzyme conformation

BIOORGANIC & MEDICINAL CHEMISTRY LETTERS 28 : 10 pp. 1693-1698. , 6 p. (2018)

DOI WoS Scopus PubMed

Publication:3375019 Validated Core Citing Journal Article (Article ) Scientific

Article (Journal Article) | Scientific[3375019] [Validated]

All citations+mentions: 5, External citations: 5, Self citations: 0, Unhandled citations: 0

Szilágyi, B. ; Ferenczy, G.G. ; Keserű, G.M. ✉

Drug discovery strategies and the preclinical development of D-amino-acid oxidase inhibitors as antipsychotic therapies

EXPERT OPINION ON DRUG DISCOVERY 13 : 10 pp. 973-982. , 10 p. (2018)

DOI WoS Scopus PubMed

Publication:30353690 Validated Core Citing Duplum Journal Article (Survey paper ) Scientific

Survey paper (Journal Article) | Scientific[30353690] [Validated]

All citations+mentions: 9, External citations: 8, Self citations: 1, Unhandled citations: 0

10.

Szilagyi, B ; Kovacs, P ; Ferenczy, GG ; Racz, A ; Nemeth, K ; Visy, J ; Szabo, P ; Ilas, J ; Balogh, GT ; Monostory, K et al.

Discovery of isatin and 1H-indazol-3-ol derivatives as d-amino acid oxidase (DAAO) inhibitors

BIOORGANIC & MEDICINAL CHEMISTRY 26 : 8 pp. 1579-1587. , 9 p. (2018)

DOI SE Repozitórium WoS Scopus PubMed Google scholar

Locked Publication:3344151 Admin approved Core Citing Journal Article (Article ) Scientific

Article (Journal Article) | Scientific[3344151] [Admin approved]

All citations+mentions: 10, External citations: 9, Self citations: 1, Unhandled citations: 0

11.

L, Somsák ; M, Polyák ; G, Varga ; J, Begum ; B, Szilágyi ; L, Juhász ; T, Docsa ; P, Gergely ; J M, Hayes

N-(β-D-Glucopyranosyl) Oxadiazole- and 1,2,4-Triazolecarboxamides as Glycogen Phosphorylase Inhibitors: Synthesis, Enzyme Kinetics and Computational Evaluation

In: 27th International Carbohydrate Symposium

Bengaluru, India : IISC (2014) Paper: I-P-58

Publication:2517810 Admin approved Core Conference paper (Abstract ) Scientific

Abstract (Conference paper) | Scientific[2517810] [Admin approved]

12.

Mária, Polyák ; Gergő, Varga ; Bence, Szilágyi ; Tibor, Docsa ; Pál, Gergely ; László, Juhász ; László, Somsák

Synthesis and enzyme kinetic evaluation of heterocyclic bioisosteric analogues of N-acyl-N’-β-D-glucopyranosyl urea type glycogen phosphorylase inhibitors

In: Ernest, Giralt (eds.) 5th European Conference on Chemistry for Life Sciences, Abstract Book

Barcelona, Spain (2013) p. 93

Publication:2382460 Admin approved Core Conference paper (Abstract ) Scientific

Abstract (Conference paper) | Scientific[2382460] [Admin approved]

13.

Polyák, M ; Varga, G ; Szilágyi, B ; Juhász, L ; Docsa, T ; Gergely, P ; Begum, J ; Hayes, JM ; Somsák, L ✉

Synthesis, enzyme kinetics and computational evaluation of N-(beta-D-glucopyranosyl) oxadiazolecarboxamides as glycogen phosphorylase inhibitors

BIOORGANIC & MEDICINAL CHEMISTRY 21 pp. 5738-5747. , 10 p. (2013)

DOI REAL WoS DEA Scopus PubMed Teljes dokumentum

Publication:2381496 Published Core Citing Journal Article (Article ) Scientific

Article (Journal Article) | Scientific[2381496] [Approved]

All citations+mentions: 23, External citations: 11, Self citations: 12, Unhandled citations: 0

14.

Polyák, Mária ; Varga, Gergely ; Szilágyi, Bence ; Docsa, Tibor ; Gergely, Pál ; Juhász, László ; Somsák, László

N-Acil-N’-β-D-glükopiranozil-karbamid típusú glikogén foszforiláz inhibitorok heterociklusos bioizosztér analógjainak szintézise és enzimkinetikai vizsgálata

In: Magyar, Kémikusok Egyesülete (eds.) Vegyészkonferencia 2013 : 2013. június 26-28., Hajdúszoboszló : program és elődásösszefoglalók

Bp, Hungary : Magyar Kémikusok Egyesülete (MKE) (2013) 152 p. p. 114 Paper: P-54

Publication:2382468 Admin approved Core Chapter in Book (Abstract ) Scientific

Abstract (Chapter in Book) | Scientific[2382468] [Admin approved]

15.

Marietta, Tóth ; Gergely, Tibor Varga ; Mária, Polyák ; Bence, Szilágyi ; Sándor, Kun ; I, Takács ; László, Juhász ; Tibor, Docsa ; Pál, Gergely ; László, Somsák

SAR study of glycogen phosphorylase inhibitors: heterocycles as bioisosteric amide replacements in N-acyl-beta-D-glucopyranosylamines and N-acyl-N’-beta-D-glucopyranosyl ureas

In: 26th International Carbohydrate Symposium

(2012) Paper: P122

Publication:2314255 Admin approved Core Conference paper (Abstract ) Scientific

Abstract (Conference paper) | Scientific[2314255] [Admin approved]

16.

Tóth, M ; Varga, G T ; Polyák, M ; Szilágyi, B ; Kun, S ; Takács, I ; Juhász, L ; Docsa, T ; Gergely, P ; Somsák, L

SAR Study of Glycogen Phosphorylase Inhibitors: Heterocycles as Bioisosteric Amide Replacements in N-Acyl-beta-D-Glucopyranosylamines and N-Acyl-N’-beta-D-Glucopyranosyl Ureas

In: 26th International Carbohydrate Symposium

(2012) pp. F80-F80.

Publication:2034044 Admin approved Core Conference paper (Abstract ) Scientific

Abstract (Conference paper) | Scientific[2034044] [Admin approved]

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