https://m2.mtmt.hu/ eng 2026-07-28 17:03 JournalArticle 34445373 VALIDATED true Medicinal Chemistry Research Group, Research Centre for Natural Sciences, Magyar tudósok krt 2, Budapest, H-1117, Hungary Department of Organic Chemistry and Technology, Faculty of Chemical Technology and Biotechnology, Budapest University of Technology and Economics, Müegyetem rkp. 3., Budapest, H-1111, Hungary National Laboratory for Drug Research and Development, Budapest, H-1117, Hungary Department of Chemical Engineering and Biotechnology, University of Applied Sciences Darmstadt, Haardtring 100, Darmstadt, 64295, Germany Institute of Animal Breeding and Genetics, University of Veterinary Medicine, Vienna, 1210, Austria MS Metabolomics Research Group, Research Centre for Natural Sciences, Magyar tudósok krt 2, Budapest, H-1117, Hungary Export Date: 14 March 2024 CODEN: JMCMA Correspondence Address: Meyer-Almes, F.-J.; Department of Chemical Engineering and Biotechnology, Haardtring 100, Germany; email: franz-josef.meyer-almes@h-da.de Correspondence Address: Keserü, G.M.; Medicinal Chemistry Research Group, Magyar tudósok krt 2, Hungary; email: keseru.gyorgy@ttk.hu 0 false 2026-07-13T14:11:48.557+0000 2025-03-27T15:18:21.792+0000 2023-12-20T11:09:52.682+0000 true 10068805 Bajusz Dávid /api/admin/10068805 Admin Dávid Bajusz (MTA TTK SZKI admin5) true 2024-11-12T15:32:57.968+0000 2024-11-12T15:32:57.968+0000 2024-02-15T11:32:07.374+0000 true 521 Szuper Admin /api/admin/521 Admin Admin Szuper (admin) true Admin 10023792 /api/admin/10023792 Margit Suchanek-Lukács (Admin 3, admin) Suchanek-Lukács Margit true 10023792 true Admin 10067876 /api/admin/10067876 Gusztáv Ladányi (MTMT API user, admin) Ladányi Gusztáv true true 2024-10-17T16:35:19.342+0000 true false true 24 24 /api/publicationtype/24 PublicationType Journal Article 1 true 24 JournalArticle true 10000059 Article true 24 24 /api/publicationtype/24 PublicationType Journal Article 1 true 24 JournalArticle /api/subtype/10000059 Szakcikk SubType Article (Journal Article) 101 true 10000059 true 1 /api/category/1 Category Scientific true 1 Keeley, Aaron B. true true /api/journal/2648 REVIEWED JOURNAL OF MEDICINAL CHEMISTRY 0022-2623 1520-4804 true false 2648 false 2648 true 0022-2623 1520-4804 Journal FOREIGN 67 1 572 585 572 14 2024 Screening of ultra-low-molecular weight ligands (MiniFrags) successfully identified viable chemical starting points for a variety of drug targets. Here we report the electrophilic analogues of MiniFrags that allow the mapping of potential binding sites for covalent inhibitors by biochemical screening and mass spectrometry. Small electrophilic heterocycles and their N-quaternized analogues were first characterized in the glutathione assay to analyze their electrophilic reactivity. Next, the library was used for systematic mapping of potential covalent binding sites available in human histone deacetylase 8 (HDAC8). The covalent labeling of HDAC8 cysteines has been proven by tandem mass spectrometry measurements, and the observations were explained by mutating HDAC8 cysteines. As a result, screening of electrophilic MiniFrags identified three potential binding sites suitable for the development of allosteric covalent HDAC8 inhibitors. One of the hit fragments was merged with a known HDAC8 inhibitor fragment using different linkers, and the linker length was optimized to result in a lead-like covalent inhibitor. © 2023 The Authors. Published by American Chemical Society Funding 2034804 /api/funding/2034804 Nemzeti Gyógyszerkutatási és Fejlesztési Laboratórium(PharmaLab) Funder: NRDIO false true true 2023 true true true false true false GOLD 2026-07-13 true https://doi.org/10.1021/acs.jmedchem.3c01779 11 0 11 8 2 11 11 11 4 11 11 8 8 8 3 0 11 8 11 8 0 7 7 Folyóiratcikk Journal Article 24 11 Könyvrészlet Chapter in Book 25 0 Könyv Book 23 0 Egyéb konferenciaközlemény Conference paper 31 0 Egyéb konferenciakötet Conference proceedings 32 0 Oltalmi formák Protection forms 26 0 Disszertáció Thesis 28 0 Egyéb Miscellaneous 29 0 Alkotás Achievement 22 0 Kutatási adat Research data 33 0 Folyóiratcikk Journal Article 24 0 0 0 Könyvrészlet Chapter in Book 25 0 0 0 Könyv Book 23 0 0 0 Egyéb konferenciaközlemény Conference paper 31 0 0 0 Egyéb konferenciakötet Conference proceedings 32 0 0 0 Oltalmi formák Protection forms 26 0 0 0 Disszertáció Thesis 28 0 0 0 Egyéb Miscellaneous 29 0 0 0 Alkotás Achievement 22 0 0 0 Kutatási adat Research data 33 0 0 0 2024 0 5 4 5 4 2025 0 4 3 4 3 2026 0 2 1 2 1 D1 false 10044995,10053848,10042926 false false false 2024-03-19T11:09:58.241+0000 Gyógyszerkémiai Kutatócsoport (HRN TTK / SZKI); Szerkezetkutató Központ (HRN TTK); Szerves Kémia és Technológia Tanszék (BME / VBK) 9 26 3 17 0 true 10023792 10067876 Language 10002 /api/language/10002 English Angol English true 2 true PersonAuthorship 113370861 /api/authorship/113370861 Keeley, Aaron B. [Keeley, Aaron Brian (kémiai tudományok), author] Gyógyszerkémiai Kutatócsoport (IOC) 1 0.059 true false false Author 10061376 /api/author/10061376 Aaron Brian Keeley (kémiai tudományok) Keeley Aaron Brian true 10061376 true Keeley Aaron B. true false false AuthorshipType 1 /api/authorshiptype/1 Author 0 true 0 true false true PersonAuthorship 113370862 /api/authorship/113370862 Kopranovic, Aleksandra 2 0.05882353 false false false Kopranovic Aleksandra true false false AuthorshipType 1 /api/authorshiptype/1 Author 0 true 0 true false true PersonAuthorship 113370863 /api/authorship/113370863 Di Lorenzo, Vincenzo [Di Lorenzo, Vincenzo (gyógyszerkémia), author] 3 0.05882353 false false false Author 10099883 /api/author/10099883 Vincenzo Di Lorenzo (gyógyszerkémia) Di Lorenzo Vincenzo true true Di Lorenzo Vincenzo true false false AuthorshipType 1 /api/authorshiptype/1 Author 0 true 0 true false true PersonAuthorship 113370864 /api/authorship/113370864 Ábrányi-Balogh, Péter [Ábrányi-Balogh, Péter (szerves kémia), author] Department of Organic Chemistry and Technology (BUTE / FCTB); Gyógyszerkémiai Kutatócsoport (IOC) 4 0.059 false false false Author 10042926 /api/author/10042926 Péter Ábrányi-Balogh (szerves kémia) Ábrányi-Balogh Péter true 10042926 true Ábrányi-Balogh Péter true false false AuthorshipType 1 /api/authorshiptype/1 Author 0 true 0 true false true PersonAuthorship 113370865 /api/authorship/113370865 Jänsch, Niklas 5 0.05882353 false false false Jänsch Niklas true false false AuthorshipType 1 /api/authorshiptype/1 Author 0 true 0 true false true PersonAuthorship 113370866 /api/authorship/113370866 Lai, Linh N. 6 0.05882353 false false false Lai Linh N. true false false AuthorshipType 1 /api/authorshiptype/1 Author 0 true 0 true false true PersonAuthorship 113370867 /api/authorship/113370867 Petri, László [Petri, László (szerves kémia, gy...), author] Gyógyszerkémiai Kutatócsoport (IOC) 7 0.059 false false false Author 10053848 /api/author/10053848 László Petri (szerves kémia, gyógyszerkémia) Petri László true 10053848 true Petri László true false false AuthorshipType 1 /api/authorshiptype/1 Author 0 true 0 true false true PersonAuthorship 113370868 /api/authorship/113370868 Orgován, Zoltán [Orgován, Zoltán (Gyógyszervegyész-...), author] Gyógyszerkémiai Kutatócsoport (IOC) 8 0.059 false false false Author 10065817 /api/author/10065817 Zoltán Orgován (Gyógyszervegyész-mérnök) Orgován Zoltán true true Orgován Zoltán true false false AuthorshipType 1 /api/authorshiptype/1 Author 0 true 0 true false true PersonAuthorship 113370869 /api/authorship/113370869 Pölöske, Daniel 9 0.05882353 false false false Pölöske Daniel true false false AuthorshipType 1 /api/authorshiptype/1 Author 0 true 0 true false true PersonAuthorship 113370870 /api/authorship/113370870 Orlova, Anna 10 0.05882353 false false false Orlova Anna true false false AuthorshipType 1 /api/authorshiptype/1 Author 0 true 0 true false true PersonAuthorship 113370871 /api/authorship/113370871 Németh, András György [Németh, András György (Szerves kémia), author] Department of Organic Chemistry and Technology (BUTE / FCTB); Gyógyszerkémiai Kutatócsoport (IOC) 11 0.059 false false false Author 10073290 /api/author/10073290 András György Németh (Szerves kémia) Németh András György true true Németh András György true false false AuthorshipType 1 /api/authorshiptype/1 Author 0 true 0 true false true PersonAuthorship 113370872 /api/authorship/113370872 Desczyk, Charlotte 12 0.05882353 false false false Desczyk Charlotte true false false AuthorshipType 1 /api/authorshiptype/1 Author 0 true 0 true false true PersonAuthorship 113370873 /api/authorship/113370873 Imre, Tímea [Imre, Timea (Tömegspektrometria), author] Centre for Structural Sciences 13 0.05882353 false false false Author 10014805 /api/author/10014805 Timea Imre (Tömegspektrometria) Imre Timea true 10014805 true Imre Tímea true false false AuthorshipType 1 /api/authorshiptype/1 Author 0 true 0 true false true PersonAuthorship 113370874 /api/authorship/113370874 Bajusz, Dávid [Bajusz, Dávid (gyógyszerkémia, m...), author] Gyógyszerkémiai Kutatócsoport (IOC) 14 0.059 false false false Author 10044995 /api/author/10044995 Dávid Bajusz (gyógyszerkémia, molekulamodellezés) Bajusz Dávid true 10044995 true Bajusz Dávid true false false AuthorshipType 1 /api/authorshiptype/1 Author 0 true 0 true false true PersonAuthorship 113370875 /api/authorship/113370875 Moriggl, Richard 15 0.05882353 false false false Moriggl Richard true false false AuthorshipType 1 /api/authorshiptype/1 Author 0 true 0 true false true PersonAuthorship 113370876 /api/authorship/113370876 Meyer-Almes, Franz-Josef 16 0.05882353 false false false Meyer-Almes Franz-Josef true false false AuthorshipType 1 /api/authorshiptype/1 Author 0 true 0 true false true PersonAuthorship 113370877 /api/authorship/113370877 Keserü, György M. ✉ [Keserű, György Miklós (Gyógyszerkémia, g...), author] Department of Organic Chemistry and Technology (BUTE / FCTB); Gyógyszerkémiai Kutatócsoport (IOC) 17 0.059 false true true Author 10001451 /api/author/10001451 György Miklós Keserű (Gyógyszerkémia, gyógyszertervezés) Keserű György Miklós true 10001451 true Keserü György M. true false false AuthorshipType 1 /api/authorshiptype/1 Author 0 true 0 true false true PublicationIdentifier 25129278 /api/publicationidentifier/25129278 DOI: 10.1021/acs.jmedchem.3c01779 PlainSource 6 /api/publicationsource/6 DOI PublicationSourceType 10001 /api/publicationsourcetype/10001 DOI true true true DOI DOI https://doi.org/@@@ true true 6 true GOLD true IDENTICAL 10.1021/acs.jmedchem.3c01779 https://doi.org/10.1021/acs.jmedchem.3c01779 false true PublicationIdentifier 25511262 /api/publicationidentifier/25511262 WoS: 001141763000001 PlainSource 1 /api/publicationsource/1 WoS PublicationSourceType 10003 /api/publicationsourcetype/10003 Indexelő adatbázis false true true WoS WoS https://www.webofscience.com/wos/woscc/full-record/@@@ true true 1 true IDENTICAL 001141763000001 https://www.webofscience.com/wos/woscc/full-record/001141763000001 false true PublicationIdentifier 29858586 /api/publicationidentifier/29858586 REAL: 224479 SwordSource 36 /api/publicationsource/36 REAL PublicationSourceType 10007 /api/publicationsourcetype/10007 Repozitórium true true true REAL REAL https://real.mtak.hu/@@@ true true 36 true GOLD true 224479 https://real.mtak.hu/224479 false true PublicationIdentifier 25279839 /api/publicationidentifier/25279839 Scopus: 85180939847 PlainSource 3 /api/publicationsource/3 Scopus PublicationSourceType 10003 /api/publicationsourcetype/10003 Indexelő adatbázis false true true Scopus Scopus http://www.scopus.com/record/display.url?origin=inward&eid=2-s2.0-@@@ true true 3 true IDENTICAL 85180939847 http://www.scopus.com/record/display.url?origin=inward&eid=2-s2.0-85180939847 false true PublicationIdentifier 25511263 /api/publicationidentifier/25511263 PubMed: 38113354 PlainSource 17 /api/publicationsource/17 PubMed PublicationSourceType 10003 /api/publicationsourcetype/10003 Indexelő adatbázis false true true PubMed PubMed http://www.ncbi.nlm.nih.gov/entrez/query.fcgi?cmd=Retrieve&db=PubMed&list_uids=@@@&dopt=Abstract true true 17 true IDENTICAL 38113354 http://www.ncbi.nlm.nih.gov/entrez/query.fcgi?cmd=Retrieve&db=PubMed&list_uids=38113354&dopt=Abstract false true PublicationIdentifier 25129279 /api/publicationidentifier/25129279 Other URL: https://pubs.acs.org/doi/10.1021/acs.jmedchem.3c01779 PlainSource 40 /api/publicationsource/40 Other URL PublicationSourceType 10006 /api/publicationsourcetype/10006 Link true true true Egyéb URL Other URL @@@ true true 40 true IDENTICAL https://pubs.acs.org/doi/10.1021/acs.jmedchem.3c01779 https://pubs.acs.org/doi/10.1021/acs.jmedchem.3c01779 false true SjrRating 11456073 /api/sjrrating/11456073 sjr:D1 (2024) Scopus - Drug Discovery JOURNAL OF MEDICINAL CHEMISTRY 0022-2623 1520-4804 11 0.1 journal RatingType 10002 /api/ratingtype/10002 sjr sjr true true ClassificationExternal 3002 /api/classificationexternal/3002 Scopus - Drug Discovery true 3002 true D1 DIRECT true true Reference 48146499 /api/reference/48146499 1. 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(2024) JOURNAL OF MEDICINAL CHEMISTRY 0022-2623 1520-4804 67 1 572-585<div class="JournalArticle Publication long-list"> <div class="authors"> <img title="Forrásközlemény" style="float: left" src="/frontend/resources/grid/publication-core-icon.png"> <img title="Idézőközlemény" style="float: left" src="/frontend/resources/grid/publication-citation-icon.png"> <div class="autype autype0"> <span class="author-name" mtid="10061376"><a href="/gui2/?type=authors&mode=browse&sel=10061376" target="_blank">Keeley Aaron B. (<span class="authorship-author-name">Keeley Aaron Brian</span> <span class="authorAux-mtmt"> kémiai tudományok</span>) </a> </span> <span class="author-affil"><span title="HUN-REN Research Centre for Natural Sciences">HUN-REN RCNS</span>/<span title="Institute of Organic Chemistry">IOC</span>/Gyógyszerkémiai Kutatócsoport</span> ;&nbsp;&nbsp;&nbsp; <span class="author-name" >Kopranovic Aleksandra </span> ;&nbsp;&nbsp;&nbsp; <span class="author-name" mtid="10099883"><a href="/gui2/?type=authors&mode=browse&sel=10099883" target="_blank">Di Lorenzo Vincenzo (<span class="authorship-author-name">Di Lorenzo Vincenzo</span> <span class="authorAux-mtmt"> gyógyszerkémia</span>) </a> </span> ;&nbsp;&nbsp;&nbsp; <span class="author-name" mtid="10042926"><a href="/gui2/?type=authors&mode=browse&sel=10042926" target="_blank">Ábrányi-Balogh Péter (<span class="authorship-author-name">Ábrányi-Balogh Péter</span> <span class="authorAux-mtmt"> szerves kémia</span>) </a> </span> <span class="author-affil"><span title="Budapest University of Technology and Economics">BUTE</span>/<span title="Faculty of Chemical Technology and Biotechnology">FCTB</span>/Department of Organic Chemistry and Technology; <span title="HUN-REN Research Centre for Natural Sciences">HUN-REN RCNS</span>/<span title="Institute of Organic Chemistry">IOC</span>/Gyógyszerkémiai Kutatócsoport</span> ;&nbsp;&nbsp;&nbsp; <span class="author-name" >Jänsch Niklas </span> ;&nbsp;&nbsp;&nbsp; <span class="author-name" >Lai Linh N. </span> ;&nbsp;&nbsp;&nbsp; <span class="author-name" mtid="10053848"><a href="/gui2/?type=authors&mode=browse&sel=10053848" target="_blank">Petri László (<span class="authorship-author-name">Petri László</span> <span class="authorAux-mtmt"> szerves kémia, gyógyszerkémia</span>) </a> </span> <span class="author-affil"><span title="HUN-REN Research Centre for Natural Sciences">HUN-REN RCNS</span>/<span title="Institute of Organic Chemistry">IOC</span>/Gyógyszerkémiai Kutatócsoport</span> ;&nbsp;&nbsp;&nbsp; <span class="author-name" mtid="10065817"><a href="/gui2/?type=authors&mode=browse&sel=10065817" target="_blank">Orgován Zoltán (<span class="authorship-author-name">Orgován Zoltán</span> <span class="authorAux-mtmt"> Gyógyszervegyész-mérnök</span>) </a> </span> <span class="author-affil"><span title="HUN-REN Research Centre for Natural Sciences">HUN-REN RCNS</span>/<span title="Institute of Organic Chemistry">IOC</span>/Gyógyszerkémiai Kutatócsoport</span> ;&nbsp;&nbsp;&nbsp; <span class="author-name" >Pölöske Daniel </span> ;&nbsp;&nbsp;&nbsp; <span class="author-name" >Orlova Anna </span> ;&nbsp;&nbsp;&nbsp; <span class="author-name" mtid="10073290"><a href="/gui2/?type=authors&mode=browse&sel=10073290" target="_blank">Németh András György (<span class="authorship-author-name">Németh András György</span> <span class="authorAux-mtmt"> Szerves kémia</span>) </a> </span> <span class="author-affil"><span title="Budapest University of Technology and Economics">BUTE</span>/<span title="Faculty of Chemical Technology and Biotechnology">FCTB</span>/Department of Organic Chemistry and Technology; <span title="HUN-REN Research Centre for Natural Sciences">HUN-REN RCNS</span>/<span title="Institute of Organic Chemistry">IOC</span>/Gyógyszerkémiai Kutatócsoport</span> ;&nbsp;&nbsp;&nbsp; <span class="author-name" >Desczyk Charlotte </span> ;&nbsp;&nbsp;&nbsp; <span class="author-name" mtid="10014805"><a href="/gui2/?type=authors&mode=browse&sel=10014805" target="_blank">Imre Tímea (<span class="authorship-author-name">Imre Timea</span> <span class="authorAux-mtmt"> Tömegspektrometria</span>) </a> </span> <span class="author-affil"><span title="HUN-REN Research Centre for Natural Sciences">HUN-REN RCNS</span>/Centre for Structural Sciences</span> ;&nbsp;&nbsp;&nbsp; <span class="author-name" mtid="10044995"><a href="/gui2/?type=authors&mode=browse&sel=10044995" target="_blank">Bajusz Dávid (<span class="authorship-author-name">Bajusz Dávid</span> <span class="authorAux-mtmt"> gyógyszerkémia, molekulamodellezés</span>) </a> </span> <span class="author-affil"><span title="HUN-REN Research Centre for Natural Sciences">HUN-REN RCNS</span>/<span title="Institute of Organic Chemistry">IOC</span>/Gyógyszerkémiai Kutatócsoport</span> ;&nbsp;&nbsp;&nbsp; <span class="author-name" >Moriggl Richard </span> ;&nbsp;&nbsp;&nbsp; <span class="author-name" >Meyer-Almes Franz-Josef </span> ;&nbsp;&nbsp;&nbsp; <span class="author-name" mtid="10001451"><a href="/gui2/?type=authors&mode=browse&sel=10001451" target="_blank">Keserü György M. ✉ (<span class="authorship-author-name">Keserű György Miklós</span> <span class="authorAux-mtmt"> Gyógyszerkémia, gyógyszertervezés</span>) </a> </span> <span class="author-affil"><span title="Budapest University of Technology and Economics">BUTE</span>/<span title="Faculty of Chemical Technology and Biotechnology">FCTB</span>/Department of Organic Chemistry and Technology; <span title="HUN-REN Research Centre for Natural Sciences">HUN-REN RCNS</span>/<span title="Institute of Organic Chemistry">IOC</span>/Gyógyszerkémiai Kutatócsoport</span> </div> </div> <div class="title"><a href="/gui2/?mode=browse&params=publication;34445373" target="_blank">Electrophilic MiniFrags Revealed Unprecedented Binding Sites for Covalent HDAC8 Inhibitors</a></div> <div> <span class="journal-title">JOURNAL OF MEDICINAL CHEMISTRY</span> <span class="journal-issn">(<a target="_blank" href="https://portal.issn.org/resource/ISSN/0022-2623">0022-2623</a> <a target="_blank" href="https://portal.issn.org/resource/ISSN/1520-4804">1520-4804</a>)</span>: <span class="journal-volume">67</span> <span class="journal-issue">1</span> <span class="page"> pp 572-585 </span> <span class="year">(2024)</span> </div> <div class="pub-footer"> <span class="language" xmlns="http://www.w3.org/1999/html">Language: English | </span> <span class="identifiers"> <span class="id identifier oa_GOLD" title=" Gold "> <a style="color:blue" title="10.1021/acs.jmedchem.3c01779" target="_blank" href="https://doi.org/10.1021/acs.jmedchem.3c01779"> DOI </a> </span> <span class="id identifier oa_none" title="none"> <a style="color:blue" title="001141763000001" target="_blank" href="https://www.webofscience.com/wos/woscc/full-record/001141763000001"> WoS </a> </span> <span class="id identifier oa_GOLD" title=" Gold "> <a style="color:black" title="224479" target="_blank" href="https://real.mtak.hu/224479"> REAL </a> </span> <span class="id identifier oa_none" title="none"> <a style="color:blue" title="85180939847" target="_blank" href="http://www.scopus.com/record/display.url?origin=inward&eid=2-s2.0-85180939847"> Scopus </a> </span> <span class="id identifier oa_none" title="none"> <a style="color:blue" title="38113354" target="_blank" href="http://www.ncbi.nlm.nih.gov/entrez/query.fcgi?cmd=Retrieve&db=PubMed&list_uids=38113354&dopt=Abstract"> PubMed </a> </span> <span class="id identifier oa_none" title="none"> <a style="color:blue" title="https://pubs.acs.org/doi/10.1021/acs.jmedchem.3c01779" target="_blank" href="https://pubs.acs.org/doi/10.1021/acs.jmedchem.3c01779"> Other URL </a> </span> </span> <OnlyViewableByAuthor><div class="ratings"> <div class="journal-subject">Journal subject: Scopus - Drug Discovery&nbsp;&nbsp;&nbsp;Rank:&nbsp;D1</div> <div class="journal-subject">Journal subject: Scopus - Molecular Medicine&nbsp;&nbsp;&nbsp;Rank:&nbsp;Q1</div> </div></OnlyViewableByAuthor> <div class="publication-citation" style="margin-left: 0.5cm;"> <span title="" class="citingPub-count">Citing papers: 11</span> | Independent citation: 8 | Self citation: 3 | Unknown citation: 0 | Number of citations in WoS: 11 | Number of citations in Scopus:&nbsp;4 | WoS/Scopus assigned:&nbsp;11 | Number of citations with DOI:&nbsp;11 </div> <div class="publication-citation"> <a target="_blank" href="/api/publication?cond=citations.related;eq;34445373&sort=publishedYear,desc&sort=title"> Number of cited publications: 7 </a> </div> <div class="mtid"><span class="long-pub-mtid">Publication: 34445373</span> | <span class="status-data status-VALIDATED"> Validated </span> Core Citing | <span class="type-subtype">Journal Article ( Article ) </span> | <span class="pub-category">Scientific</span> | <span class="publication-sourceOfData">kézi felvitel</span> </div> <div class="funder"> Nemzeti Gyógyszerkutatási és Fejlesztési Laboratórium (PharmaLab)(RRF-2.3.1-21-2022-00015) Funder: NRDIO </div> <div class="lastModified">Last Modified: 2025.03.27. 16:18 Dávid Bajusz (MTA TTK SZKI admin5) </div> <div class="lockedBy">Centrally managed 2024.10.17. 18:35 Margit Suchanek-Lukács (Admin 3, admin) Gusztáv Ladányi (MTMT API user, admin) </div> <pre class="comment" style="margin-top: 0; margin-bottom: 0;"><u>Comments</u>: Medicinal Chemistry Research Group, Research Centre for Natural Sciences, Magyar tudósok krt 2, Budapest, H-1117, Hungary Department of Organic Chemistry and Technology, Faculty of Chemical Technology and Biotechnology, Budapest University of Technology and Economics, Müegyetem rkp. 3., Budapest, H-1111, Hungary National Laboratory for Drug Resear...</pre> </div></div>